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A first-in-man phase 1 study of the DNA-dependent protein kinase inhibitor peposertib (formerly M3814) in patients with advanced solid tumours.
van Bussel, Mark T J; Awada, Ahmad; de Jonge, Maja J A; Mau-Sørensen, Morten; Nielsen, Dorte; Schöffski, Patrick; Verheul, Henk M W; Sarholz, Barbara; Berghoff, Karin; El Bawab, Samer; Kuipers, Mirjam; Damstrup, Lars; Diaz-Padilla, Ivan; Schellens, Jan H M.
Afiliação
  • van Bussel MTJ; Department of Clinical Pharmacology, The Netherlands Cancer Institute, Amsterdam, The Netherlands. m.v.bussel@nki.nl.
  • Awada A; Oncology Medicine Department, Jules Bordet Institute, Université Libre de Bruxelles, Brussels, Belgium.
  • de Jonge MJA; Medical Oncology, Erasmus MC Cancer Institute, Rotterdam, The Netherlands.
  • Mau-Sørensen M; Department of Oncology, Rigshospitalet, Copenhagen, Denmark.
  • Nielsen D; Department of Oncology, Herlev and Gentofte Hospital, Herlev, Denmark.
  • Schöffski P; Department of General Medical Oncology, Leuven Cancer Institute, University Hospitals Leuven, Leuven, Belgium.
  • Verheul HMW; Department of Medical Oncology, Radboud University Medical Center, Nijmegen, The Netherlands.
  • Sarholz B; Merck KGaA, Darmstadt, Germany.
  • Berghoff K; Merck KGaA, Darmstadt, Germany.
  • El Bawab S; Merck KGaA, Darmstadt, Germany.
  • Kuipers M; Merck KGaA, Darmstadt, Germany.
  • Damstrup L; Merck KGaA, Darmstadt, Germany.
  • Diaz-Padilla I; Debiopharm International S.A., Lausanne, Switzerland.
  • Schellens JHM; Ares Trading S.A., Eysins, Switzerland; an Affiliate of Merck KGaA, Darmstadt, Germany.
Br J Cancer ; 124(4): 728-735, 2021 02.
Article em En | MEDLINE | ID: mdl-33230210

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Piridazinas / Quinazolinas / Proteína Quinase Ativada por DNA / Neoplasias Idioma: En Ano de publicação: 2021 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Piridazinas / Quinazolinas / Proteína Quinase Ativada por DNA / Neoplasias Idioma: En Ano de publicação: 2021 Tipo de documento: Article