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The CUL3/neddylation inhibitor MLN4924 reduces ethanol-induced locomotor sensitization and inflammatory pain allodynia in mice.
Ding, Zhong; Knipp, Gregory T; van Rijn, Richard M; Chester, Julia A; Watts, Val J.
Afiliação
  • Ding Z; Dept of Medicinal Chemistry & Molecular Pharmacology, Purdue University, West Lafayette, IN, 47907, USA.
  • Knipp GT; Dept of Industrial and Physical Pharmacy, Purdue University, West Lafayette, IN, 47907, USA; Purdue Institute for Drug Discovery, Purdue University, West Lafayette, IN, 47907, USA.
  • van Rijn RM; Dept of Medicinal Chemistry & Molecular Pharmacology, Purdue University, West Lafayette, IN, 47907, USA; Purdue Institute for Drug Discovery, Purdue University, West Lafayette, IN, 47907, USA; Purdue Institute for Integrative Neuroscience, Purdue University, West Lafayette, IN, 47907, USA.
  • Chester JA; Purdue Institute for Integrative Neuroscience, Purdue University, West Lafayette, IN, 47907, USA; Dept of Psychological Sciences, Purdue University, West Lafayette, IN, 47907, USA.
  • Watts VJ; Dept of Medicinal Chemistry & Molecular Pharmacology, Purdue University, West Lafayette, IN, 47907, USA; Purdue Institute for Drug Discovery, Purdue University, West Lafayette, IN, 47907, USA; Purdue Institute for Integrative Neuroscience, Purdue University, West Lafayette, IN, 47907, USA. Elect
Behav Brain Res ; 399: 113051, 2021 02 05.
Article em En | MEDLINE | ID: mdl-33279641

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Pirimidinas / Depressores do Sistema Nervoso Central / Ciclopentanos / Proteínas Culina / Etanol / Alcoolismo / Inibidores Enzimáticos / Sensibilização do Sistema Nervoso Central / Proteína NEDD8 / Hiperalgesia Idioma: En Ano de publicação: 2021 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Pirimidinas / Depressores do Sistema Nervoso Central / Ciclopentanos / Proteínas Culina / Etanol / Alcoolismo / Inibidores Enzimáticos / Sensibilização do Sistema Nervoso Central / Proteína NEDD8 / Hiperalgesia Idioma: En Ano de publicação: 2021 Tipo de documento: Article