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A broad-spectrum substrate for the human UDP-glucuronosyltransferases and its use for investigating glucuronidation inhibitors.
Zhou, Qi-Hang; Qin, Wei-Wei; Finel, Moshe; He, Qing-Qing; Tu, Dong-Zhu; Wang, Chao-Ran; Ge, Guang-Bo.
Afiliação
  • Zhou QH; Institute of Interdisciplinary Integrative Medicine Research, Shanghai University of Traditional Chinese Medicine, Shanghai 201203, China.
  • Qin WW; Department of Pharmacy, Huashan Hospital, Fudan University, Shanghai 200040, China.
  • Finel M; Division of Pharmaceutical Chemistry and Technology, Faculty of Pharmacy, University of Helsinki, 00014, Finland.
  • He QQ; Institute of Interdisciplinary Integrative Medicine Research, Shanghai University of Traditional Chinese Medicine, Shanghai 201203, China.
  • Tu DZ; Institute of Interdisciplinary Integrative Medicine Research, Shanghai University of Traditional Chinese Medicine, Shanghai 201203, China.
  • Wang CR; Dalian Institute of Chemical Physics, Chinese Academy of Sciences, Dalian 116023, China.
  • Ge GB; Institute of Interdisciplinary Integrative Medicine Research, Shanghai University of Traditional Chinese Medicine, Shanghai 201203, China. Electronic address: geguangbo@dicp.ac.cn.
Int J Biol Macromol ; 180: 252-261, 2021 Jun 01.
Article em En | MEDLINE | ID: mdl-33741369

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Glucuronosiltransferase / Inibidores Enzimáticos / Benzodioxóis / Isoflavonas Idioma: En Ano de publicação: 2021 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Glucuronosiltransferase / Inibidores Enzimáticos / Benzodioxóis / Isoflavonas Idioma: En Ano de publicação: 2021 Tipo de documento: Article