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Identification of positive modulators of TRPM5 channel from a high-throughput screen using a fluorescent membrane potential assay.
Virginio, Caterina; Aldegheri, Laura; Nola, Selena; Brodbeck, Daniela; Brault, Laurent; Raveglia, Luca F; Barilli, Alessio; Sabat, Mark; Myers, Richard.
Afiliação
  • Virginio C; Aptuit, an Evotec Company, Via Alessandro Fleming, 4, 37135 Verona, Italy. Electronic address: caterina.virginio@evotec.com.
  • Aldegheri L; Aptuit, an Evotec Company, Via Alessandro Fleming, 4, 37135 Verona, Italy.
  • Nola S; Aptuit, an Evotec Company, Via Alessandro Fleming, 4, 37135 Verona, Italy.
  • Brodbeck D; Aptuit, an Evotec Company, Via Alessandro Fleming, 4, 37135 Verona, Italy.
  • Brault L; Aptuit, an Evotec Company, Via Alessandro Fleming, 4, 37135 Verona, Italy.
  • Raveglia LF; Aptuit, an Evotec Company, Via Alessandro Fleming, 4, 37135 Verona, Italy.
  • Barilli A; Aptuit, an Evotec Company, Via Alessandro Fleming, 4, 37135 Verona, Italy.
  • Sabat M; Takeda Pharmaceuticals, 9625 Towne Centre Drive, San Diego, CA 92121, United States.
  • Myers R; Takeda Pharmaceuticals, 9625 Towne Centre Drive, San Diego, CA 92121, United States.
SLAS Discov ; 27(1): 55-64, 2022 01.
Article em En | MEDLINE | ID: mdl-35058176

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Canais de Potencial de Receptor Transitório / Canais de Cátion TRPM Idioma: En Ano de publicação: 2022 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Canais de Potencial de Receptor Transitório / Canais de Cátion TRPM Idioma: En Ano de publicação: 2022 Tipo de documento: Article