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Identification of non-ATP-competitive α-carboline inhibitors of the anaplastic lymphoma kinase.
Mologni, Luca; Orsato, Alexandre; Zambon, Alfonso; Tardy, Sébastien; Bisson, William H; Schneider, Cedric; Ceccon, Monica; Viltadi, Michela; D'Attoma, Joseph; Pannilunghi, Sara; Vece, Vito; Gueyrard, David; Bertho, Jerome; Scapozza, Leonardo; Goekjian, Peter; Gambacorti-Passerini, Carlo.
Afiliação
  • Mologni L; Dept. of Medicine and Surgery, University of Milano-Bicocca, Monza, Italy; Galkem Srl, Monza, Italy. Electronic address: luca.mologni@unimib.it.
  • Orsato A; Laboratoire Chimie Organique 2-Glycochimie, CNRS-Université Claude Bernard Lyon 1, Villeurbanne, France; Dept. of Chemistry, Universidade Estadual de Londrina, Paraná, Brazil.
  • Zambon A; Department of Chemistry and Geological Sciences, University of Modena and Reggio Emilia, Modena, Italy.
  • Tardy S; Laboratoire Chimie Organique 2-Glycochimie, CNRS-Université Claude Bernard Lyon 1, Villeurbanne, France; School of Pharmaceutical Sciences, University of Geneva, Switzerland; Institute of Pharmaceutical Sciences of Western Switzerland, University of Geneva, Switzerland.
  • Bisson WH; School of Pharmaceutical Sciences, University of Geneva, Switzerland; Knight Cancer Institute, Oregon Health & Science University, Portland, OR, USA.
  • Schneider C; Laboratoire Chimie Organique 2-Glycochimie, CNRS-Université Claude Bernard Lyon 1, Villeurbanne, France.
  • Ceccon M; Dept. of Medicine and Surgery, University of Milano-Bicocca, Monza, Italy.
  • Viltadi M; Dept. of Medicine and Surgery, University of Milano-Bicocca, Monza, Italy.
  • D'Attoma J; Laboratoire Chimie Organique 2-Glycochimie, CNRS-Université Claude Bernard Lyon 1, Villeurbanne, France.
  • Pannilunghi S; School of Pharmaceutical Sciences, University of Geneva, Switzerland; Institute of Pharmaceutical Sciences of Western Switzerland, University of Geneva, Switzerland.
  • Vece V; Dept. of Medicine and Surgery, University of Milano-Bicocca, Monza, Italy; Department of Chemistry, Massachusetts Institute of Technology, Cambridge, MA, USA.
  • Gueyrard D; Laboratoire Chimie Organique 2-Glycochimie, CNRS-Université Claude Bernard Lyon 1, Villeurbanne, France.
  • Bertho J; Galkem Srl, Monza, Italy.
  • Scapozza L; Galkem Srl, Monza, Italy; School of Pharmaceutical Sciences, University of Geneva, Switzerland; Institute of Pharmaceutical Sciences of Western Switzerland, University of Geneva, Switzerland. Electronic address: leonardo.scapozza@unige.ch.
  • Goekjian P; Galkem Srl, Monza, Italy; Laboratoire Chimie Organique 2-Glycochimie, CNRS-Université Claude Bernard Lyon 1, Villeurbanne, France.
  • Gambacorti-Passerini C; Dept. of Medicine and Surgery, University of Milano-Bicocca, Monza, Italy; Galkem Srl, Monza, Italy.
Eur J Med Chem ; 238: 114488, 2022 Aug 05.
Article em En | MEDLINE | ID: mdl-35665691

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Carbolinas / Receptores Proteína Tirosina Quinases Idioma: En Ano de publicação: 2022 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Carbolinas / Receptores Proteína Tirosina Quinases Idioma: En Ano de publicação: 2022 Tipo de documento: Article