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Design, synthesis and biological evaluation of novel osimertinib derivatives as reversible EGFR kinase inhibitors.
Ding, Shi; Gao, Ziye; Hu, Ziqiang; Qi, Rui; Zheng, Xiangshan; Dong, Xiaoyong; Zhang, Mingjuan; Shen, Jiwei; Long, Tian; Zhu, Yan; Tian, Lu; Song, Wenshan; Liu, Ruoqing; Li, Ying; Sun, Jiahuan; Duan, Wenwen; Liu, Ju; Chen, Ye.
Afiliação
  • Ding S; College of Pharmacy of Liaoning University, 66 Chongshan Road, Huanggu District, Shenyang, 110036, PR China; API Engineering Technology Research Center of Liaoning Province, 66 Chongshan Road, Huanggu District, Shenyang, 110036, PR China; Small Molecular Targeted Drug R&D Engineering Research Ce
  • Gao Z; College of Pharmacy of Liaoning University, 66 Chongshan Road, Huanggu District, Shenyang, 110036, PR China.
  • Hu Z; College of Pharmacy of Liaoning University, 66 Chongshan Road, Huanggu District, Shenyang, 110036, PR China.
  • Qi R; College of Pharmacy of Liaoning University, 66 Chongshan Road, Huanggu District, Shenyang, 110036, PR China.
  • Zheng X; College of Pharmacy of Liaoning University, 66 Chongshan Road, Huanggu District, Shenyang, 110036, PR China.
  • Dong X; College of Pharmacy of Liaoning University, 66 Chongshan Road, Huanggu District, Shenyang, 110036, PR China.
  • Zhang M; College of Pharmacy of Liaoning University, 66 Chongshan Road, Huanggu District, Shenyang, 110036, PR China.
  • Shen J; College of Pharmacy of Liaoning University, 66 Chongshan Road, Huanggu District, Shenyang, 110036, PR China; API Engineering Technology Research Center of Liaoning Province, 66 Chongshan Road, Huanggu District, Shenyang, 110036, PR China; Small Molecular Targeted Drug R&D Engineering Research Ce
  • Long T; College of Pharmacy of Liaoning University, 66 Chongshan Road, Huanggu District, Shenyang, 110036, PR China.
  • Zhu Y; College of Pharmacy of Liaoning University, 66 Chongshan Road, Huanggu District, Shenyang, 110036, PR China.
  • Tian L; College of Pharmacy of Liaoning University, 66 Chongshan Road, Huanggu District, Shenyang, 110036, PR China.
  • Song W; College of Pharmacy of Liaoning University, 66 Chongshan Road, Huanggu District, Shenyang, 110036, PR China.
  • Liu R; College of Pharmacy of Liaoning University, 66 Chongshan Road, Huanggu District, Shenyang, 110036, PR China.
  • Li Y; College of Pharmacy of Liaoning University, 66 Chongshan Road, Huanggu District, Shenyang, 110036, PR China.
  • Sun J; College of Pharmacy of Liaoning University, 66 Chongshan Road, Huanggu District, Shenyang, 110036, PR China.
  • Duan W; IHuman Institute, ShanghaiTech University, 393 Middle Huaxia Road, Pudong District, Shanghai, 201210, PR China.
  • Liu J; College of Pharmacy of Liaoning University, 66 Chongshan Road, Huanggu District, Shenyang, 110036, PR China; API Engineering Technology Research Center of Liaoning Province, 66 Chongshan Road, Huanggu District, Shenyang, 110036, PR China; Small Molecular Targeted Drug R&D Engineering Research Ce
  • Chen Y; College of Pharmacy of Liaoning University, 66 Chongshan Road, Huanggu District, Shenyang, 110036, PR China; API Engineering Technology Research Center of Liaoning Province, 66 Chongshan Road, Huanggu District, Shenyang, 110036, PR China; Small Molecular Targeted Drug R&D Engineering Research Ce
Eur J Med Chem ; 238: 114492, 2022 Aug 05.
Article em En | MEDLINE | ID: mdl-35696862

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Carcinoma Pulmonar de Células não Pequenas / Neoplasias Pulmonares Idioma: En Ano de publicação: 2022 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Carcinoma Pulmonar de Células não Pequenas / Neoplasias Pulmonares Idioma: En Ano de publicação: 2022 Tipo de documento: Article