A 'click' chemistry approach to novel entinostat (MS-275) based class I histone deacetylase proteolysis targeting chimeras.

Cross, Jasmine M; Coulson, Megan E; Smalley, Joshua P; Pytel, Wiktoria A; Ismail, Ozair; Trory, Justin S; Cowley, Shaun M; Hodgkinson, James T.

Afiliação

Cross JM; Leicester Institute of Structural and Chemical Biology, School of Chemistry, University of Leicester Leicester LE1 7RH UK JTHodgkinson@le.ac.uk.
Coulson ME; Leicester Institute of Structural and Chemical Biology, School of Chemistry, University of Leicester Leicester LE1 7RH UK JTHodgkinson@le.ac.uk.
Smalley JP; Department of Molecular and Cell Biology, University of Leicester Leicester LE1 7RH UK smc57@leicester.ac.uk.
Pytel WA; Leicester Institute of Structural and Chemical Biology, School of Chemistry, University of Leicester Leicester LE1 7RH UK JTHodgkinson@le.ac.uk.
Ismail O; Leicester Institute of Structural and Chemical Biology, School of Chemistry, University of Leicester Leicester LE1 7RH UK JTHodgkinson@le.ac.uk.
Trory JS; Department of Molecular and Cell Biology, University of Leicester Leicester LE1 7RH UK smc57@leicester.ac.uk.
Cowley SM; Leicester Institute of Structural and Chemical Biology, School of Chemistry, University of Leicester Leicester LE1 7RH UK JTHodgkinson@le.ac.uk.
Hodgkinson JT; Leicester Institute of Structural and Chemical Biology, School of Chemistry, University of Leicester Leicester LE1 7RH UK JTHodgkinson@le.ac.uk.

RSC Med Chem ; 13(12): 1634-1639, 2022 Dec 14.

Article em En | MEDLINE | ID: mdl-36545434

Texto completo: 1 Base de dados: MEDLINE Idioma: En Ano de publicação: 2022 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Idioma: En Ano de publicação: 2022 Tipo de documento: Article