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Discovery of potent 1,1-diarylthiogalactoside glycomimetic inhibitors of Pseudomonas aeruginosa LecA with antibiofilm properties.
Bruneau, Alexandre; Gillon, Emilie; Furiga, Aurélie; Brachet, Etienne; Alami, Mouad; Roques, Christine; Varrot, Annabelle; Imberty, Anne; Messaoudi, Samir.
Afiliação
  • Bruneau A; BioCIS, Univ. Paris-Sud, CNRS, University Paris-Saclay, Châtenay-Malabry, France.
  • Gillon E; Université Grenoble Alpes, CNRS, CERMAV, 38000, Grenoble, France.
  • Furiga A; LCG, Laboratoire de Génie Chimique (UMR 5503), Département Bioprocédés et Systèmes Microbiens, Université de Toulouse, CNRS, INPT, UPS, Toulouse, France.
  • Brachet E; BioCIS, Univ. Paris-Sud, CNRS, University Paris-Saclay, Châtenay-Malabry, France.
  • Alami M; BioCIS, Univ. Paris-Sud, CNRS, University Paris-Saclay, Châtenay-Malabry, France.
  • Roques C; LCG, Laboratoire de Génie Chimique (UMR 5503), Département Bioprocédés et Systèmes Microbiens, Université de Toulouse, CNRS, INPT, UPS, Toulouse, France.
  • Varrot A; Université Grenoble Alpes, CNRS, CERMAV, 38000, Grenoble, France.
  • Imberty A; Université Grenoble Alpes, CNRS, CERMAV, 38000, Grenoble, France. Electronic address: anne.imberty@cermav.cnrs.fr.
  • Messaoudi S; BioCIS, Univ. Paris-Sud, CNRS, University Paris-Saclay, Châtenay-Malabry, France. Electronic address: samir.messaoudi@universite-paris-saclay.fr.
Eur J Med Chem ; 247: 115025, 2023 Feb 05.
Article em En | MEDLINE | ID: mdl-36549118

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Pseudomonas aeruginosa / Adesinas Bacterianas Idioma: En Ano de publicação: 2023 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Pseudomonas aeruginosa / Adesinas Bacterianas Idioma: En Ano de publicação: 2023 Tipo de documento: Article