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"Hit" to lead optimization and chemoinformatic studies for a new series of Autotaxin inhibitors.
Stylianaki, Elli-Anna; Magkrioti, Christiana; Ladopoulou, Eleni M; Papavasileiou, Konstantinos D; Lagarias, Panagiotis; Melagraki, Georgia; Samiotaki, Martina; Panayotou, George; Dedos, Skarlatos G; Afantitis, Antreas; Aidinis, Vassilis; Matralis, Alexios N.
Afiliação
  • Stylianaki EA; Bioinnovation Institute, Biomedical Sciences Research Center "Alexander Fleming, Athens, Greece.
  • Magkrioti C; Bioinnovation Institute, Biomedical Sciences Research Center "Alexander Fleming, Athens, Greece.
  • Ladopoulou EM; Bioinnovation Institute, Biomedical Sciences Research Center "Alexander Fleming, Athens, Greece; Department of Biology, National and Kapodistrian University of Athens, Zografou, Athens, Greece.
  • Papavasileiou KD; NovaMechanics Ltd, Larnaca, Cyprus; NovaMechanics MIKE, Piraeus, Greece.
  • Lagarias P; NovaMechanics Ltd, Larnaca, Cyprus.
  • Melagraki G; Division of Physical Sciences and Applications, Hellenic Military Academy, Vari, Greece.
  • Samiotaki M; Bioinnovation Institute, Biomedical Sciences Research Center "Alexander Fleming, Athens, Greece.
  • Panayotou G; Bioinnovation Institute, Biomedical Sciences Research Center "Alexander Fleming, Athens, Greece.
  • Dedos SG; Department of Biology, National and Kapodistrian University of Athens, Zografou, Athens, Greece.
  • Afantitis A; NovaMechanics Ltd, Larnaca, Cyprus; NovaMechanics MIKE, Piraeus, Greece. Electronic address: afantitis@novamechanics.com.
  • Aidinis V; Bioinnovation Institute, Biomedical Sciences Research Center "Alexander Fleming, Athens, Greece. Electronic address: aidinis@fleming.gr.
  • Matralis AN; Bioinnovation Institute, Biomedical Sciences Research Center "Alexander Fleming, Athens, Greece. Electronic address: matralis@fleming.gr.
Eur J Med Chem ; 249: 115130, 2023 Mar 05.
Article em En | MEDLINE | ID: mdl-36702053

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Fibrose Pulmonar Idiopática / Neoplasias Idioma: En Ano de publicação: 2023 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Fibrose Pulmonar Idiopática / Neoplasias Idioma: En Ano de publicação: 2023 Tipo de documento: Article