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Going beyond Binary: Rapid Identification of Protein-Protein Interaction Modulators Using a Multifragment Kinetic Target-Guided Synthesis Approach.
Nacheva, Katya; Kulkarni, Sameer S; Kassu, Mintesinot; Flanigan, David; Monastyrskyi, Andrii; Iyamu, Iredia D; Doi, Kenichiro; Barber, Megan; Namelikonda, Niranjan; Tipton, Jeremiah D; Parvatkar, Prakash; Wang, Hong-Gang; Manetsch, Roman.
Afiliação
  • Nacheva K; Department of Chemistry, University of South Florida, Tampa, Florida 33620, United States.
  • Kulkarni SS; Department of Chemistry, University of South Florida, Tampa, Florida 33620, United States.
  • Kassu M; Department of Chemistry and Chemical Biology, Northeastern University, Boston, Massachusetts 02115, United States.
  • Flanigan D; Department of Chemistry, University of South Florida, Tampa, Florida 33620, United States.
  • Monastyrskyi A; Department of Sciences, Hillsborough Community College, Tampa, Florida 33619, United States.
  • Iyamu ID; Department of Chemistry, University of South Florida, Tampa, Florida 33620, United States.
  • Doi K; Department of Chemistry, University of South Florida, Tampa, Florida 33620, United States.
  • Barber M; Department of Chemistry and Chemical Biology, Northeastern University, Boston, Massachusetts 02115, United States.
  • Namelikonda N; Department of Pediatrics, Division of Pediatric Hematology and Oncology, Penn State College of Medicine, Hershey, Pennsylvania 17033, United States.
  • Tipton JD; Department of Chemistry, University of South Florida, Tampa, Florida 33620, United States.
  • Parvatkar P; Department of Chemistry, University of South Florida, Tampa, Florida 33620, United States.
  • Wang HG; Proteomics and Mass Spectrometry Core Facility, University of South Florida, Tampa, Florida 33620, United States.
  • Manetsch R; Department of Chemistry and Chemical Biology, Northeastern University, Boston, Massachusetts 02115, United States.
J Med Chem ; 66(7): 5196-5207, 2023 04 13.
Article em En | MEDLINE | ID: mdl-37000900

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Descoberta de Drogas Idioma: En Ano de publicação: 2023 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Descoberta de Drogas Idioma: En Ano de publicação: 2023 Tipo de documento: Article