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Identification of novel class inhibitors of NSD3 methyltransferase showing a unique, bivalent binding mode in the SET domain.
Kim, Sumin; Hwang, Injeoung; Kim, Suhn Hyung; Chung, Hwan Won; Ji, Mi-Jung; Moon, Sojeong; Park, Hyun-Mee; Kong, Gu; Hur, Wooyoung.
Afiliação
  • Kim S; HY-KIST Bioconvergence, Hanyang University, Seoul, South Korea.
  • Hwang I; HY-KIST Bioconvergence, Hanyang University, Seoul, South Korea.
  • Kim SH; Medicinal Materials Research Center, Korea Institute of Science and Technology (KIST), Seoul, South Korea.
  • Chung HW; Medicinal Materials Research Center, Korea Institute of Science and Technology (KIST), Seoul, South Korea.
  • Ji MJ; Computational Science Research Center, Korea Institute of Science and Technology (KIST), Seoul, South Korea.
  • Moon S; Advanced Analysis Data Center, Korea Institute of Science and Technology (KIST), Seoul, South Korea.
  • Park HM; HY-KIST Bioconvergence, Hanyang University, Seoul, South Korea.
  • Kong G; Advanced Analysis Data Center, Korea Institute of Science and Technology (KIST), Seoul, South Korea.
  • Hur W; HY-KIST Bioconvergence, Hanyang University, Seoul, South Korea.
Chem Biol Drug Des ; 102(3): 500-513, 2023 09.
Article em En | MEDLINE | ID: mdl-37072259

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Neoplasias da Mama / Domínios PR-SET Idioma: En Ano de publicação: 2023 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Neoplasias da Mama / Domínios PR-SET Idioma: En Ano de publicação: 2023 Tipo de documento: Article