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Discovery of a Novel Series of Potent SHP2 Allosteric Inhibitors.
Petrocchi, Alessia; Grillo, Alessandro; Ferrante, Luca; Randazzo, Pietro; Prandi, Adolfo; De Matteo, Marilenia; Iaccarino, Costanza; Bisbocci, Monica; Cellucci, Antonella; Alli, Cristina; Nibbio, Martina; Pucci, Vincenzo; Amaudrut, Jérôme; Montalbetti, Christian; Toniatti, Carlo; Di Fabio, Romano.
Afiliação
  • Petrocchi A; IRBM S.p.A, Via Pontina Km 30.600, 00070 Pomezia, Italy.
  • Grillo A; Promidis, Via Olgettina 60, 20132 Milano, Italy.
  • Ferrante L; Promidis, Via Olgettina 60, 20132 Milano, Italy.
  • Randazzo P; Promidis, Via Olgettina 60, 20132 Milano, Italy.
  • Prandi A; Promidis, Via Olgettina 60, 20132 Milano, Italy.
  • De Matteo M; Promidis, Via Olgettina 60, 20132 Milano, Italy.
  • Iaccarino C; IRBM S.p.A, Via Pontina Km 30.600, 00070 Pomezia, Italy.
  • Bisbocci M; IRBM S.p.A, Via Pontina Km 30.600, 00070 Pomezia, Italy.
  • Cellucci A; IRBM S.p.A, Via Pontina Km 30.600, 00070 Pomezia, Italy.
  • Alli C; IRBM S.p.A, Via Pontina Km 30.600, 00070 Pomezia, Italy.
  • Nibbio M; IRBM S.p.A, Via Pontina Km 30.600, 00070 Pomezia, Italy.
  • Pucci V; IRBM S.p.A, Via Pontina Km 30.600, 00070 Pomezia, Italy.
  • Amaudrut J; IRBM S.p.A, Via Pontina Km 30.600, 00070 Pomezia, Italy.
  • Montalbetti C; IRBM S.p.A, Via Pontina Km 30.600, 00070 Pomezia, Italy.
  • Toniatti C; IRBM S.p.A, Via Pontina Km 30.600, 00070 Pomezia, Italy.
  • Di Fabio R; IRBM S.p.A, Via Pontina Km 30.600, 00070 Pomezia, Italy.
ACS Med Chem Lett ; 14(5): 645-651, 2023 May 11.
Article em En | MEDLINE | ID: mdl-37197453

Texto completo: 1 Base de dados: MEDLINE Idioma: En Ano de publicação: 2023 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Idioma: En Ano de publicação: 2023 Tipo de documento: Article