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Structure-Based Design and Synthesis of Stapled 10Panx1 Analogues for Use in Cardiovascular Inflammatory Diseases.
Lamouroux, Arthur; Tournier, Malaury; Iaculli, Debora; Caufriez, Anne; Rusiecka, Olga M; Martin, Charlotte; Bes, Viviane; Carpio, Laureano E; Girardin, Yana; Loris, Remy; Tabernilla, Andrés; Molica, Filippo; Gozalbes, Rafael; Mayán, María D; Vinken, Mathieu; Kwak, Brenda R; Ballet, Steven.
Afiliação
  • Lamouroux A; Research Group of Organic Chemistry, Departments of Chemistry and Bioengineering Sciences, Vrije Universiteit Brussel, Pleinlaan 2, B-1050 Brussels, Belgium.
  • Tournier M; Department of Pathology and Immunology and Geneva Center for Inflammation Research, Faculty of Medicine, University of Geneva, Rue Michel-Servet 1, CH-1211 Geneva, Switzerland.
  • Iaculli D; Research Group of Organic Chemistry, Departments of Chemistry and Bioengineering Sciences, Vrije Universiteit Brussel, Pleinlaan 2, B-1050 Brussels, Belgium.
  • Caufriez A; Research Group of Organic Chemistry, Departments of Chemistry and Bioengineering Sciences, Vrije Universiteit Brussel, Pleinlaan 2, B-1050 Brussels, Belgium.
  • Rusiecka OM; Research Unit of In Vitro Toxicology and Dermato-Cosmetology, Department of Pharmaceutical Sciences, Vrije Universiteit Brussel, Laarbeeklaan 103, 1090 Brussels, Belgium.
  • Martin C; Department of Pathology and Immunology and Geneva Center for Inflammation Research, Faculty of Medicine, University of Geneva, Rue Michel-Servet 1, CH-1211 Geneva, Switzerland.
  • Bes V; Research Group of Organic Chemistry, Departments of Chemistry and Bioengineering Sciences, Vrije Universiteit Brussel, Pleinlaan 2, B-1050 Brussels, Belgium.
  • Carpio LE; Department of Pathology and Immunology and Geneva Center for Inflammation Research, Faculty of Medicine, University of Geneva, Rue Michel-Servet 1, CH-1211 Geneva, Switzerland.
  • Girardin Y; ProtoQSAR SL, Centro Europeo de Empresas Innovadoras, Parque Tecnológico de Valencia, Avda. Benjamin Franklin 12, 46980 Paterna, Spain.
  • Loris R; Structural Biology Brussels, Department of Biotechnology, Vrije Universiteit Brussel, Pleinlaan 2, B-1050 Brussels, Belgium.
  • Tabernilla A; Centre for Structural Biology, VIB, Pleinlaan 2, 1050 Brussels, Belgium.
  • Molica F; Structural Biology Brussels, Department of Biotechnology, Vrije Universiteit Brussel, Pleinlaan 2, B-1050 Brussels, Belgium.
  • Gozalbes R; Centre for Structural Biology, VIB, Pleinlaan 2, 1050 Brussels, Belgium.
  • Mayán MD; Research Unit of In Vitro Toxicology and Dermato-Cosmetology, Department of Pharmaceutical Sciences, Vrije Universiteit Brussel, Laarbeeklaan 103, 1090 Brussels, Belgium.
  • Vinken M; Department of Pathology and Immunology and Geneva Center for Inflammation Research, Faculty of Medicine, University of Geneva, Rue Michel-Servet 1, CH-1211 Geneva, Switzerland.
  • Kwak BR; ProtoQSAR SL, Centro Europeo de Empresas Innovadoras, Parque Tecnológico de Valencia, Avda. Benjamin Franklin 12, 46980 Paterna, Spain.
  • Ballet S; MolDrug AI Systems SL, c/Olimpia Arozena 45, 46018 Valencia, Spain.
J Med Chem ; 66(18): 13086-13102, 2023 09 28.
Article em En | MEDLINE | ID: mdl-37703077

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Doenças Cardiovasculares / Conexinas Idioma: En Ano de publicação: 2023 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Doenças Cardiovasculares / Conexinas Idioma: En Ano de publicação: 2023 Tipo de documento: Article