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Small Molecule Ligands of the BET-like Bromodomain, SmBRD3, Affect Schistosoma mansoni Survival, Oviposition, and Development.
Schiedel, Matthias; McArdle, Darius J B; Padalino, Gilda; Chan, Anthony K N; Forde-Thomas, Josephine; McDonough, Michael; Whiteland, Helen; Beckmann, Manfred; Cookson, Rosa; Hoffmann, Karl F; Conway, Stuart J.
Afiliação
  • Schiedel M; Department of Chemistry, Chemistry Research Laboratory, University of Oxford, Mansfield Road, Oxford OX1 3TA, U.K.
  • McArdle DJB; Department of Chemistry, Chemistry Research Laboratory, University of Oxford, Mansfield Road, Oxford OX1 3TA, U.K.
  • Padalino G; The Department of Life Sciences (DLS), Aberystwyth University, Wales SY23 3DA, U.K.
  • Chan AKN; Department of Chemistry, Chemistry Research Laboratory, University of Oxford, Mansfield Road, Oxford OX1 3TA, U.K.
  • Forde-Thomas J; The Department of Life Sciences (DLS), Aberystwyth University, Wales SY23 3DA, U.K.
  • McDonough M; Department of Chemistry, Chemistry Research Laboratory, University of Oxford, Mansfield Road, Oxford OX1 3TA, U.K.
  • Whiteland H; The Department of Life Sciences (DLS), Aberystwyth University, Wales SY23 3DA, U.K.
  • Beckmann M; The Department of Life Sciences (DLS), Aberystwyth University, Wales SY23 3DA, U.K.
  • Cookson R; GlaxoSmithKline R&D, Stevenage, Hertfordshire SG1 2NY, U.K.
  • Hoffmann KF; The Department of Life Sciences (DLS), Aberystwyth University, Wales SY23 3DA, U.K.
  • Conway SJ; Department of Chemistry, Chemistry Research Laboratory, University of Oxford, Mansfield Road, Oxford OX1 3TA, U.K.
J Med Chem ; 66(23): 15801-15822, 2023 12 14.
Article em En | MEDLINE | ID: mdl-38048437

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Esquistossomose / Esquistossomose mansoni Idioma: En Ano de publicação: 2023 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Esquistossomose / Esquistossomose mansoni Idioma: En Ano de publicação: 2023 Tipo de documento: Article