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1.
Hit-to-lead optimization and kinase selectivity of imidazo[1,2-a]quinoxalin-4-amine derived JNK1 inhibitors.
Bioorg Med Chem Lett
; 23(18): 5217-22, 2013 Sep 15.
Article
in English
| MEDLINE | ID: mdl-23916259
2.
6-Position optimization of tricyclic 4-quinolone-based inhibitors of glycogen synthase kinase-3ß: discovery of nitrile derivatives with picomolar potency.
Bioorg Med Chem Lett
; 22(2): 1005-8, 2012 Jan 15.
Article
in English
| MEDLINE | ID: mdl-22202172
3.
Synthesis and structure-activity relationship of 4-quinolone-3-carboxylic acid based inhibitors of glycogen synthase kinase-3ß.
Bioorg Med Chem Lett
; 21(19): 5948-51, 2011 Oct 01.
Article
in English
| MEDLINE | ID: mdl-21873061
4.
Functional interrogation of the kinome using nucleotide acyl phosphates.
Biochemistry
; 46(2): 350-8, 2007 Jan 16.
Article
in English
| MEDLINE | ID: mdl-17209545
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