Detalhe da pesquisa
1.
Discovery of a novel potent GABA(B) receptor agonist.
Bioorg Med Chem Lett
; 21(21): 6582-5, 2011 Nov 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-21920749
2.
Arbaclofen placarbil, a novel R-baclofen prodrug: improved absorption, distribution, metabolism, and elimination properties compared with R-baclofen.
J Pharmacol Exp Ther
; 330(3): 911-21, 2009 Sep.
Artigo
em Inglês
| MEDLINE | ID: mdl-19502531
3.
XP13512 [(+/-)-1-([(alpha-isobutanoyloxyethoxy)carbonyl] aminomethyl)-1-cyclohexane acetic acid], a novel gabapentin prodrug: II. Improved oral bioavailability, dose proportionality, and colonic absorption compared with gabapentin in rats and monkeys.
J Pharmacol Exp Ther
; 311(1): 324-33, 2004 Oct.
Artigo
em Inglês
| MEDLINE | ID: mdl-15146029