1.
Bioorg Med Chem Lett
; 19(15): 4280-3, 2009 Aug 01.
Artigo
em Inglês
| MEDLINE
| ID: mdl-19515558
RESUMO
A series of potent Cathepsin L inhibitors with good selectivity with respect to other cysteine Cathepsins is described and SAR is discussed with reference to the crystal structure of a protein-ligand complex.