Detalhe da pesquisa
1.
Suppression of lipopolysaccharide-induced COX-2 expression via p38MAPK, JNK, and C/EBPß phosphorylation inhibition by furomagydarin A, a benzofuran glycoside from Magydaris pastinacea.
J Enzyme Inhib Med Chem
; 39(1): 2287420, 2024 Dec.
Artigo
em Inglês
| MEDLINE | ID: mdl-38058285
2.
2H-chromene and 7H-furo-chromene derivatives selectively inhibit tumour associated human carbonic anhydrase IX and XII isoforms.
J Enzyme Inhib Med Chem
; 38(1): 2270183, 2023 Dec.
Artigo
em Inglês
| MEDLINE | ID: mdl-37870190
3.
Flavonoids and Acid-Hydrolysis derivatives of Neo-Clerodane diterpenes from Teucrium flavum subsp. glaucum as inhibitors of the HIV-1 reverse transcriptase-associated RNase H function.
J Enzyme Inhib Med Chem
; 36(1): 749-757, 2021 Dec.
Artigo
em Inglês
| MEDLINE | ID: mdl-33715562
4.
Selective inhibition of carbonic anhydrase IX and XII by coumarin and psoralen derivatives.
J Enzyme Inhib Med Chem
; 36(1): 685-692, 2021 Dec.
Artigo
em Inglês
| MEDLINE | ID: mdl-33602041
5.
2-(2-Methyl-2-nitrovinyl)furan but Not Furvina Interfere with Staphylococcus aureus Agr Quorum-Sensing System and Potentiate the Action of Fusidic Acid against Biofilms.
Int J Mol Sci
; 22(2)2021 Jan 09.
Artigo
em Inglês
| MEDLINE | ID: mdl-33435417
6.
Exploring New Scaffolds for the Dual Inhibition of HIV-1 RT Polymerase and Ribonuclease Associated Functions.
Molecules
; 26(13)2021 Jun 23.
Artigo
em Inglês
| MEDLINE | ID: mdl-34201561
7.
Quercetin Blocks Ebola Virus Infection by Counteracting the VP24 Interferon-Inhibitory Function.
Antimicrob Agents Chemother
; 64(7)2020 06 23.
Artigo
em Inglês
| MEDLINE | ID: mdl-32366711
8.
Coumarins from Magydaris pastinacea as inhibitors of the tumour-associated carbonic anhydrases IX and XII: isolation, biological studies and in silico evaluation.
J Enzyme Inhib Med Chem
; 35(1): 539-548, 2020 Dec.
Artigo
em Inglês
| MEDLINE | ID: mdl-31948300
9.
Ferulic Acid Esters and Withanolides: In Search of Withania somnifera GABAA Receptor Modulators.
J Nat Prod
; 82(5): 1250-1257, 2019 05 24.
Artigo
em Inglês
| MEDLINE | ID: mdl-30998355
10.
Exploring new structural features of the 4-[(3-methyl-4-aryl-2,3-dihydro-1,3-thiazol-2-ylidene)amino]benzenesulphonamide scaffold for the inhibition of human carbonic anhydrases.
J Enzyme Inhib Med Chem
; 34(1): 1526-1533, 2019 Dec.
Artigo
em Inglês
| MEDLINE | ID: mdl-31431095
11.
From cycloheptathiophene-3-carboxamide to oxazinone-based derivatives as allosteric HIV-1 ribonuclease H inhibitors.
J Enzyme Inhib Med Chem
; 34(1): 55-74, 2019 Dec.
Artigo
em Inglês
| MEDLINE | ID: mdl-30362381
12.
Identification of Myricetin as an Ebola Virus VP35-Double-Stranded RNA Interaction Inhibitor through a Novel Fluorescence-Based Assay.
Biochemistry
; 57(44): 6367-6378, 2018 11 06.
Artigo
em Inglês
| MEDLINE | ID: mdl-30298725
13.
Identification of G-quadruplex DNA/RNA binders: Structure-based virtual screening and biophysical characterization.
Biochim Biophys Acta Gen Subj
; 1861(5 Pt B): 1329-1340, 2017 May.
Artigo
em Inglês
| MEDLINE | ID: mdl-28025082
14.
Phenylpropenoids from Bupleurum fruticosum as Anti-Human Rhinovirus Species A Selective Capsid Binders.
J Nat Prod
; 80(10): 2799-2806, 2017 10 27.
Artigo
em Inglês
| MEDLINE | ID: mdl-29039946
15.
Isatin thiazoline hybrids as dual inhibitors of HIV-1 reverse transcriptase.
J Enzyme Inhib Med Chem
; 32(1): 130-136, 2017 Dec.
Artigo
em Inglês
| MEDLINE | ID: mdl-27766892
16.
Through scaffold modification to 3,5-diaryl-4,5-dihydroisoxazoles: new potent and selective inhibitors of monoamine oxidase B.
J Enzyme Inhib Med Chem
; 32(1): 264-270, 2017 Dec.
Artigo
em Inglês
| MEDLINE | ID: mdl-28097874
17.
Isatin: a privileged scaffold for the design of carbonic anhydrase inhibitors.
J Enzyme Inhib Med Chem
; 32(1): 68-73, 2017 Dec.
Artigo
em Inglês
| MEDLINE | ID: mdl-27775452
18.
Exploring the thiazole scaffold for the identification of new agents for the treatment of fluconazole resistant Candida.
J Enzyme Inhib Med Chem
; 31(6): 1672-7, 2016 Dec.
Artigo
em Inglês
| MEDLINE | ID: mdl-26745285
19.
New 4-[(3-cyclohexyl-4-aryl-2,3-dihydro-1,3-thiazol-2-ylidene)amino]benzene-1-sulfonamides, synthesis and inhibitory activity toward carbonic anhydrase I, II, IX, XII.
Bioorg Med Chem Lett
; 25(16): 3281-4, 2015 Aug 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-26073006
20.
Methoxyflavones from Stachys glutinosa with binding affinity to opioid receptors: in silico, in vitro, and in vivo studies.
J Nat Prod
; 78(1): 69-76, 2015 Jan 23.
Artigo
em Inglês
| MEDLINE | ID: mdl-25562563