Detalhe da pesquisa
1.
Substituted benzyloxytricyclic compounds as retinoic acid-related orphan receptor gamma t (RORγt) agonists.
Bioorg Med Chem Lett
; 30(12): 127204, 2020 06 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-32334911
2.
Discovery of hydroxyl 1,2-diphenylethanamine analogs as potent cholesterol ester transfer protein inhibitors.
Bioorg Med Chem Lett
; 26(14): 3278-3281, 2016 07 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-27256912
3.
Diphenylpyridylethanamine (DPPE)-based aminoheterocycles as cholesteryl ester transfer protein inhibitors.
Bioorg Med Chem Lett
; 24(3): 860-4, 2014 Feb 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-24424134
4.
Identification of a potent and metabolically stable series of fluorinated diphenylpyridylethanamine-based cholesteryl ester transfer protein inhibitors.
Bioorg Med Chem Lett
; 22(20): 6503-8, 2012 Oct 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-22995620
5.
Pyrrolo[1,2-f]triazines as JAK2 inhibitors: achieving potency and selectivity for JAK2 over JAK3.
Bioorg Med Chem Lett
; 21(5): 1425-8, 2011 Mar 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-21282055
6.
Discovery and Preclinical Pharmacology of an Oral Bromodomain and Extra-Terminal (BET) Inhibitor Using Scaffold-Hopping and Structure-Guided Drug Design.
J Med Chem
; 64(19): 14247-14265, 2021 10 14.
Artigo
em Inglês
| MEDLINE | ID: mdl-34543572
7.
Design and synthesis of a G-protein-coupled receptor antagonist library of aryloxyalkanolamines using a polymer-supported acyclic acetal linker.
J Comb Chem
; 11(1): 72-82, 2009.
Artigo
em Inglês
| MEDLINE | ID: mdl-19086798
8.
Discovery of a Lead Triphenylethanamine Cholesterol Ester Transfer Protein (CETP) Inhibitor.
ACS Med Chem Lett
; 10(6): 911-916, 2019 Jun 13.
Artigo
em Inglês
| MEDLINE | ID: mdl-31223447
9.
2-Arylbenzoxazoles as novel cholesteryl ester transfer protein inhibitors: optimization via array synthesis.
Bioorg Med Chem Lett
; 18(8): 2640-4, 2008 Apr 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-18374566
10.
Triphenylethanamine Derivatives as Cholesteryl Ester Transfer Protein Inhibitors: Discovery of N-[(1R)-1-(3-Cyclopropoxy-4-fluorophenyl)-1-[3-fluoro-5-(1,1,2,2-tetrafluoroethoxy)phenyl]-2-phenylethyl]-4-fluoro-3-(trifluoromethyl)benzamide (BMS-795311).
J Med Chem
; 58(22): 9010-26, 2015 Nov 25.
Artigo
em Inglês
| MEDLINE | ID: mdl-26524347
11.
Diphenylpyridylethanamine (DPPE) derivatives as cholesteryl ester transfer protein (CETP) inhibitors.
J Med Chem
; 55(13): 6162-75, 2012 Jul 12.
Artigo
em Inglês
| MEDLINE | ID: mdl-22650305
12.
Solid-phase synthesis of 5-substituted amino pyrazoles.
J Comb Chem
; 7(4): 584-8, 2005.
Artigo
em Inglês
| MEDLINE | ID: mdl-16004502
13.
3-Azido-3-deoxy-glycopyranoside derivatives as scaffolds for the synthesis of carbohydrate-based universal pharmacophore mapping libraries.
Bioorg Med Chem Lett
; 13(13): 2185-9, 2003 Jul 07.
Artigo
em Inglês
| MEDLINE | ID: mdl-12798331