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Biochemical Screening of Five Protein Kinases from Plasmodium falciparum against 14,000 Cell-Active Compounds.
Crowther, Gregory J; Hillesland, Heidi K; Keyloun, Katelyn R; Reid, Molly C; Lafuente-Monasterio, Maria Jose; Ghidelli-Disse, Sonja; Leonard, Stephen E; He, Panqing; Jones, Jackson C; Krahn, Mallory M; Mo, Jack S; Dasari, Kartheek S; Fox, Anna M W; Boesche, Markus; El Bakkouri, Majida; Rivas, Kasey L; Leroy, Didier; Hui, Raymond; Drewes, Gerard; Maly, Dustin J; Van Voorhis, Wesley C; Ojo, Kayode K.
Affiliation
  • Crowther GJ; Division of Allergy & Infectious Diseases, Department of Medicine, University of Washington, Seattle, Washington, United States of America.
  • Hillesland HK; Division of Allergy & Infectious Diseases, Department of Medicine, University of Washington, Seattle, Washington, United States of America.
  • Keyloun KR; Division of Allergy & Infectious Diseases, Department of Medicine, University of Washington, Seattle, Washington, United States of America.
  • Reid MC; Division of Allergy & Infectious Diseases, Department of Medicine, University of Washington, Seattle, Washington, United States of America.
  • Lafuente-Monasterio MJ; Tres Cantos Medicines Development Campus, GlaxoSmithKline, Tres Cantos, Madrid, Spain.
  • Ghidelli-Disse S; Cellzome GmbH, Molecular Discovery Research, GlaxoSmithKline R&D, Heidelberg, Germany.
  • Leonard SE; Department of Chemistry, University of Washington, Seattle, Washington, United States of America.
  • He P; Division of Allergy & Infectious Diseases, Department of Medicine, University of Washington, Seattle, Washington, United States of America.
  • Jones JC; Division of Allergy & Infectious Diseases, Department of Medicine, University of Washington, Seattle, Washington, United States of America.
  • Krahn MM; Division of Allergy & Infectious Diseases, Department of Medicine, University of Washington, Seattle, Washington, United States of America.
  • Mo JS; Division of Allergy & Infectious Diseases, Department of Medicine, University of Washington, Seattle, Washington, United States of America.
  • Dasari KS; Division of Allergy & Infectious Diseases, Department of Medicine, University of Washington, Seattle, Washington, United States of America.
  • Fox AM; Division of Allergy & Infectious Diseases, Department of Medicine, University of Washington, Seattle, Washington, United States of America.
  • Boesche M; Cellzome GmbH, Molecular Discovery Research, GlaxoSmithKline R&D, Heidelberg, Germany.
  • El Bakkouri M; Structural Genomics Consortium, University of Toronto, Toronto, Ontario, Canada.
  • Rivas KL; Division of Allergy & Infectious Diseases, Department of Medicine, University of Washington, Seattle, Washington, United States of America.
  • Leroy D; Drug Discovery, Medicines for Malaria Venture, Geneva, Switzerland.
  • Hui R; Structural Genomics Consortium, University of Toronto, Toronto, Ontario, Canada.
  • Drewes G; Cellzome GmbH, Molecular Discovery Research, GlaxoSmithKline R&D, Heidelberg, Germany.
  • Maly DJ; Department of Chemistry, University of Washington, Seattle, Washington, United States of America.
  • Van Voorhis WC; Division of Allergy & Infectious Diseases, Department of Medicine, University of Washington, Seattle, Washington, United States of America.
  • Ojo KK; Division of Allergy & Infectious Diseases, Department of Medicine, University of Washington, Seattle, Washington, United States of America.
PLoS One ; 11(3): e0149996, 2016.
Article in En | MEDLINE | ID: mdl-26934697

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Plasmodium falciparum / Protein Kinases / Antimalarials Type of study: Diagnostic_studies / Screening_studies Limits: Humans Language: En Journal: PLoS One Journal subject: CIENCIA / MEDICINA Year: 2016 Type: Article Affiliation country: United States

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Plasmodium falciparum / Protein Kinases / Antimalarials Type of study: Diagnostic_studies / Screening_studies Limits: Humans Language: En Journal: PLoS One Journal subject: CIENCIA / MEDICINA Year: 2016 Type: Article Affiliation country: United States