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Structure-activity relationship of a novel series of inhibitors for cancer type transporter L-type amino acid transporter 1 (LAT1).
Kongpracha, Pornparn; Nagamori, Shushi; Wiriyasermkul, Pattama; Tanaka, Yoko; Kaneda, Kazuko; Okuda, Suguru; Ohgaki, Ryuichi; Kanai, Yoshikatsu.
Affiliation
  • Kongpracha P; Department of Bio-system Pharmacology, Graduate School of Medicine, Osaka University, 2-2 Yamadaoka, Suita, Osaka 565-0871, Japan.
  • Nagamori S; Department of Bio-system Pharmacology, Graduate School of Medicine, Osaka University, 2-2 Yamadaoka, Suita, Osaka 565-0871, Japan.
  • Wiriyasermkul P; Department of Psychiatry, Columbia University College of Physicians and Surgeons, New York, NY 10032, USA.
  • Tanaka Y; Department of Bio-system Pharmacology, Graduate School of Medicine, Osaka University, 2-2 Yamadaoka, Suita, Osaka 565-0871, Japan.
  • Kaneda K; Department of Bio-system Pharmacology, Graduate School of Medicine, Osaka University, 2-2 Yamadaoka, Suita, Osaka 565-0871, Japan.
  • Okuda S; Department of Bio-system Pharmacology, Graduate School of Medicine, Osaka University, 2-2 Yamadaoka, Suita, Osaka 565-0871, Japan.
  • Ohgaki R; Department of Bio-system Pharmacology, Graduate School of Medicine, Osaka University, 2-2 Yamadaoka, Suita, Osaka 565-0871, Japan.
  • Kanai Y; Department of Bio-system Pharmacology, Graduate School of Medicine, Osaka University, 2-2 Yamadaoka, Suita, Osaka 565-0871, Japan. Electronic address: ykanai@pharma1.med.osaka-u.ac.jp.
J Pharmacol Sci ; 133(2): 96-102, 2017 Feb.
Article in En | MEDLINE | ID: mdl-28242177

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Triiodothyronine / Large Neutral Amino Acid-Transporter 1 Limits: Humans Language: En Journal: J Pharmacol Sci Journal subject: FARMACOLOGIA Year: 2017 Type: Article Affiliation country: Japan

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Triiodothyronine / Large Neutral Amino Acid-Transporter 1 Limits: Humans Language: En Journal: J Pharmacol Sci Journal subject: FARMACOLOGIA Year: 2017 Type: Article Affiliation country: Japan