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New TRAP1 and Hsp90 chaperone inhibitors with cationic components: Preliminary studies on mitochondrial targeting.
Rondanin, R; Lettini, G; Oliva, P; Baruchello, R; Costantini, C; Trapella, C; Simoni, D; Bernardi, T; Sisinni, L; Pietrafesa, M; Ponterini, G; Costi, M P; Vignudelli, T; Luciani, R; Matassa, D S; Esposito, F; Landriscina, M.
Affiliation
  • Rondanin R; Dep. of Chemical and Pharmaceutical Sciences, University of Ferrara, Italy.
  • Lettini G; Laboratory of Pre-Clinical and Translational Research, IRCCS, Referral Cancer Center of Basilicata, Rionero in Vulture, Italy.
  • Oliva P; Dep. of Chemical and Pharmaceutical Sciences, University of Ferrara, Italy.
  • Baruchello R; Dep. of Chemical and Pharmaceutical Sciences, University of Ferrara, Italy.
  • Costantini C; Dep. of Chemical and Pharmaceutical Sciences, University of Ferrara, Italy.
  • Trapella C; Dep. of Chemical and Pharmaceutical Sciences, University of Ferrara, Italy.
  • Simoni D; Dep. of Chemical and Pharmaceutical Sciences, University of Ferrara, Italy.
  • Bernardi T; Dep. of Chemical and Pharmaceutical Sciences, University of Ferrara, Italy.
  • Sisinni L; Laboratory of Pre-Clinical and Translational Research, IRCCS, Referral Cancer Center of Basilicata, Rionero in Vulture, Italy.
  • Pietrafesa M; Laboratory of Pre-Clinical and Translational Research, IRCCS, Referral Cancer Center of Basilicata, Rionero in Vulture, Italy.
  • Ponterini G; Dep. of Life Sciences, University of Modena and Reggio Emilia, Italy.
  • Costi MP; Dep. of Life Sciences, University of Modena and Reggio Emilia, Italy.
  • Vignudelli T; Dep. of Life Sciences, University of Modena and Reggio Emilia, Italy.
  • Luciani R; Dep. of Life Sciences, University of Modena and Reggio Emilia, Italy.
  • Matassa DS; Dep. of Molecular Medicine and Medical Biotechnology, University of Napoli Federico II, Italy.
  • Esposito F; Dep. of Molecular Medicine and Medical Biotechnology, University of Napoli Federico II, Italy. Electronic address: franca.esposito@unina.it.
  • Landriscina M; Laboratory of Pre-Clinical and Translational Research, IRCCS, Referral Cancer Center of Basilicata, Rionero in Vulture, Italy; Dep. of Medical and Surgical Sciences, University of Foggia, Italy. Electronic address: matteo.landriscina@unifg.it.
Bioorg Med Chem Lett ; 28(13): 2289-2293, 2018 07 15.
Article in En | MEDLINE | ID: mdl-29807796

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: HSP90 Heat-Shock Proteins / Isoxazoles / Mitochondria Limits: Humans Language: En Journal: Bioorg Med Chem Lett Journal subject: BIOQUIMICA / QUIMICA Year: 2018 Type: Article Affiliation country: Italy

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: HSP90 Heat-Shock Proteins / Isoxazoles / Mitochondria Limits: Humans Language: En Journal: Bioorg Med Chem Lett Journal subject: BIOQUIMICA / QUIMICA Year: 2018 Type: Article Affiliation country: Italy