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The KN-93 Molecule Inhibits Calcium/Calmodulin-Dependent Protein Kinase II (CaMKII) Activity by Binding to Ca2+/CaM.
Wong, Melanie H; Samal, Alexandra B; Lee, Mike; Vlach, Jiri; Novikov, Nikolai; Niedziela-Majka, Anita; Feng, Joy Y; Koltun, Dmitry O; Brendza, Katherine M; Kwon, Hyock Joo; Schultz, Brian E; Sakowicz, Roman; Saad, Jamil S; Papalia, Giuseppe A.
Affiliation
  • Wong MH; Gilead Sciences Inc, 333 Lakeside Drive, Foster City, CA 94404, USA.
  • Samal AB; Department of Microbiology, University of Alabama at Birmingham, Birmingham, AL 35294, USA.
  • Lee M; Gilead Sciences Inc, 333 Lakeside Drive, Foster City, CA 94404, USA.
  • Vlach J; Department of Microbiology, University of Alabama at Birmingham, Birmingham, AL 35294, USA.
  • Novikov N; Gilead Sciences Inc, 333 Lakeside Drive, Foster City, CA 94404, USA.
  • Niedziela-Majka A; Gilead Sciences Inc, 333 Lakeside Drive, Foster City, CA 94404, USA.
  • Feng JY; Gilead Sciences Inc, 333 Lakeside Drive, Foster City, CA 94404, USA.
  • Koltun DO; Gilead Sciences Inc, 333 Lakeside Drive, Foster City, CA 94404, USA.
  • Brendza KM; Gilead Sciences Inc, 333 Lakeside Drive, Foster City, CA 94404, USA.
  • Kwon HJ; Gilead Sciences Inc, 333 Lakeside Drive, Foster City, CA 94404, USA.
  • Schultz BE; Gilead Sciences Inc, 333 Lakeside Drive, Foster City, CA 94404, USA.
  • Sakowicz R; Gilead Sciences Inc, 333 Lakeside Drive, Foster City, CA 94404, USA.
  • Saad JS; Department of Microbiology, University of Alabama at Birmingham, Birmingham, AL 35294, USA. Electronic address: saad@uab.edu.
  • Papalia GA; Gilead Sciences Inc, 333 Lakeside Drive, Foster City, CA 94404, USA. Electronic address: jpapalia@gilead.com.
J Mol Biol ; 431(7): 1440-1459, 2019 03 29.
Article in En | MEDLINE | ID: mdl-30753871

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Sulfonamides / Benzylamines / Calmodulin / Calcium / Calcium-Calmodulin-Dependent Protein Kinase Type 2 Limits: Humans Language: En Journal: J Mol Biol Year: 2019 Type: Article Affiliation country: United States

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Sulfonamides / Benzylamines / Calmodulin / Calcium / Calcium-Calmodulin-Dependent Protein Kinase Type 2 Limits: Humans Language: En Journal: J Mol Biol Year: 2019 Type: Article Affiliation country: United States