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Protein surface topography as a tool to enhance the selective activity of a potassium channel blocker.
Berkut, Antonina A; Chugunov, Anton O; Mineev, Konstantin S; Peigneur, Steve; Tabakmakher, Valentin M; Krylov, Nikolay A; Oparin, Peter B; Lihonosova, Alyona F; Novikova, Ekaterina V; Arseniev, Alexander S; Grishin, Eugene V; Tytgat, Jan; Efremov, Roman G; Vassilevski, Alexander A.
Affiliation
  • Berkut AA; M.M. Shemyakin & Yu.A. Ovchinnikov Institute of Bioorganic Chemistry, Russian Academy of Sciences, 117997 Moscow, Russia.
  • Chugunov AO; M.M. Shemyakin & Yu.A. Ovchinnikov Institute of Bioorganic Chemistry, Russian Academy of Sciences, 117997 Moscow, Russia; National Research University Higher School of Economics, 101000 Moscow, Russia; Moscow Institute of Physics and Technology (State University), 141700 Dolgoprudny, Russia.
  • Mineev KS; M.M. Shemyakin & Yu.A. Ovchinnikov Institute of Bioorganic Chemistry, Russian Academy of Sciences, 117997 Moscow, Russia; Moscow Institute of Physics and Technology (State University), 141700 Dolgoprudny, Russia.
  • Peigneur S; Toxicology and Pharmacology, University of Leuven, 3000 Leuven, Belgium.
  • Tabakmakher VM; M.M. Shemyakin & Yu.A. Ovchinnikov Institute of Bioorganic Chemistry, Russian Academy of Sciences, 117997 Moscow, Russia; School of Biomedicine, Far Eastern Federal University, 690950 Vladivostok, Russia.
  • Krylov NA; M.M. Shemyakin & Yu.A. Ovchinnikov Institute of Bioorganic Chemistry, Russian Academy of Sciences, 117997 Moscow, Russia; National Research University Higher School of Economics, 101000 Moscow, Russia.
  • Oparin PB; M.M. Shemyakin & Yu.A. Ovchinnikov Institute of Bioorganic Chemistry, Russian Academy of Sciences, 117997 Moscow, Russia.
  • Lihonosova AF; National Research University Higher School of Economics, 101000 Moscow, Russia.
  • Novikova EV; M.M. Shemyakin & Yu.A. Ovchinnikov Institute of Bioorganic Chemistry, Russian Academy of Sciences, 117997 Moscow, Russia; Moscow Institute of Physics and Technology (State University), 141700 Dolgoprudny, Russia.
  • Arseniev AS; M.M. Shemyakin & Yu.A. Ovchinnikov Institute of Bioorganic Chemistry, Russian Academy of Sciences, 117997 Moscow, Russia; Moscow Institute of Physics and Technology (State University), 141700 Dolgoprudny, Russia.
  • Grishin EV; M.M. Shemyakin & Yu.A. Ovchinnikov Institute of Bioorganic Chemistry, Russian Academy of Sciences, 117997 Moscow, Russia.
  • Tytgat J; Toxicology and Pharmacology, University of Leuven, 3000 Leuven, Belgium.
  • Efremov RG; M.M. Shemyakin & Yu.A. Ovchinnikov Institute of Bioorganic Chemistry, Russian Academy of Sciences, 117997 Moscow, Russia; National Research University Higher School of Economics, 101000 Moscow, Russia; Moscow Institute of Physics and Technology (State University), 141700 Dolgoprudny, Russia. Ele
  • Vassilevski AA; M.M. Shemyakin & Yu.A. Ovchinnikov Institute of Bioorganic Chemistry, Russian Academy of Sciences, 117997 Moscow, Russia; Moscow Institute of Physics and Technology (State University), 141700 Dolgoprudny, Russia. Electronic address: avas@ibch.ru.
J Biol Chem ; 294(48): 18349-18359, 2019 11 29.
Article in En | MEDLINE | ID: mdl-31533989

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Peptides / Proteins / Potassium Channel Blockers / Kv1.3 Potassium Channel Limits: Animals / Humans Language: En Journal: J Biol Chem Year: 2019 Type: Article Affiliation country: RUSSIA

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Peptides / Proteins / Potassium Channel Blockers / Kv1.3 Potassium Channel Limits: Animals / Humans Language: En Journal: J Biol Chem Year: 2019 Type: Article Affiliation country: RUSSIA