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Structure-activity relationship of 4-azaindole-2-piperidine derivatives as agents against Trypanosoma cruzi.
Koovits, Paul J; Dessoy, Marco A; Matheeussen, An; Maes, Louis; Caljon, Guy; Mowbray, Charles E; Kratz, Jadel M; Dias, Luiz C.
Affiliation
  • Koovits PJ; Institute of Chemistry, University of Campinas (UNICAMP), Rua Josué de Castro, S/N, Cidade Universitária, Campinas, SP 13083-861, Brazil.
  • Dessoy MA; Institute of Chemistry, University of Campinas (UNICAMP), Rua Josué de Castro, S/N, Cidade Universitária, Campinas, SP 13083-861, Brazil.
  • Matheeussen A; Laboratory of Microbiology, Parasitology and Hygiene (LMPH), Universiteitsplein 1, 2610 Antwerpen, Belgium.
  • Maes L; Laboratory of Microbiology, Parasitology and Hygiene (LMPH), Universiteitsplein 1, 2610 Antwerpen, Belgium.
  • Caljon G; Laboratory of Microbiology, Parasitology and Hygiene (LMPH), Universiteitsplein 1, 2610 Antwerpen, Belgium.
  • Mowbray CE; Drugs for Neglected Diseases Initiative (DNDi), 15 Chemin Louis-Dunant, 1202 Geneva, Switzerland.
  • Kratz JM; Drugs for Neglected Diseases Initiative (DNDi), 15 Chemin Louis-Dunant, 1202 Geneva, Switzerland.
  • Dias LC; Institute of Chemistry, University of Campinas (UNICAMP), Rua Josué de Castro, S/N, Cidade Universitária, Campinas, SP 13083-861, Brazil. Electronic address: ldias@iqm.unicamp.br.
Bioorg Med Chem Lett ; 30(1): 126779, 2020 01 01.
Article in En | MEDLINE | ID: mdl-31706667

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Piperidines / Trypanosoma cruzi / Chagas Disease Limits: Animals / Humans Language: En Journal: Bioorg Med Chem Lett Journal subject: BIOQUIMICA / QUIMICA Year: 2020 Type: Article Affiliation country: Brazil

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Piperidines / Trypanosoma cruzi / Chagas Disease Limits: Animals / Humans Language: En Journal: Bioorg Med Chem Lett Journal subject: BIOQUIMICA / QUIMICA Year: 2020 Type: Article Affiliation country: Brazil