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Discovery of Potent and Selective MTH1 Inhibitors for Oncology: Enabling Rapid Target (In)Validation.
Farand, Julie; Kropf, Jeffrey E; Blomgren, Peter; Xu, Jianjun; Schmitt, Aaron C; Newby, Zachary E; Wang, Ting; Murakami, Eisuke; Barauskas, Ona; Sudhamsu, Jawahar; Feng, Joy Y; Niedziela-Majka, Anita; Schultz, Brian E; Schwartz, Karen; Viatchenko-Karpinski, Serge; Kornyeyev, Dmytro; Kashishian, Adam; Fan, Peidong; Chen, Xiaowu; Lansdon, Eric B; Ports, Michael O; Currie, Kevin S; Watkins, William J; Notte, Gregory T.
Affiliation
  • Farand J; Gilead Sciences, Inc. 333 Lakeside Drive, Foster City, California 94404, United States.
  • Kropf JE; Gilead Sciences, Inc. 199 East Blaine Street, Seattle, Washington 98102, United States.
  • Blomgren P; Gilead Sciences, Inc. 199 East Blaine Street, Seattle, Washington 98102, United States.
  • Xu J; Gilead Sciences, Inc. 199 East Blaine Street, Seattle, Washington 98102, United States.
  • Schmitt AC; Gilead Sciences, Inc. 199 East Blaine Street, Seattle, Washington 98102, United States.
  • Newby ZE; Gilead Sciences, Inc. 333 Lakeside Drive, Foster City, California 94404, United States.
  • Wang T; Gilead Sciences, Inc. 333 Lakeside Drive, Foster City, California 94404, United States.
  • Murakami E; Gilead Sciences, Inc. 333 Lakeside Drive, Foster City, California 94404, United States.
  • Barauskas O; Gilead Sciences, Inc. 333 Lakeside Drive, Foster City, California 94404, United States.
  • Sudhamsu J; Gilead Sciences, Inc. 333 Lakeside Drive, Foster City, California 94404, United States.
  • Feng JY; Gilead Sciences, Inc. 333 Lakeside Drive, Foster City, California 94404, United States.
  • Niedziela-Majka A; Gilead Sciences, Inc. 333 Lakeside Drive, Foster City, California 94404, United States.
  • Schultz BE; Gilead Sciences, Inc. 333 Lakeside Drive, Foster City, California 94404, United States.
  • Schwartz K; Gilead Sciences, Inc. 333 Lakeside Drive, Foster City, California 94404, United States.
  • Viatchenko-Karpinski S; Gilead Sciences, Inc. 333 Lakeside Drive, Foster City, California 94404, United States.
  • Kornyeyev D; Gilead Sciences, Inc. 333 Lakeside Drive, Foster City, California 94404, United States.
  • Kashishian A; Gilead Sciences, Inc. 199 East Blaine Street, Seattle, Washington 98102, United States.
  • Fan P; Gilead Sciences, Inc. 333 Lakeside Drive, Foster City, California 94404, United States.
  • Chen X; Gilead Sciences, Inc. 333 Lakeside Drive, Foster City, California 94404, United States.
  • Lansdon EB; Gilead Sciences, Inc. 333 Lakeside Drive, Foster City, California 94404, United States.
  • Ports MO; Gilead Sciences, Inc. 199 East Blaine Street, Seattle, Washington 98102, United States.
  • Currie KS; Gilead Sciences, Inc. 199 East Blaine Street, Seattle, Washington 98102, United States.
  • Watkins WJ; Gilead Sciences, Inc. 333 Lakeside Drive, Foster City, California 94404, United States.
  • Notte GT; Gilead Sciences, Inc. 333 Lakeside Drive, Foster City, California 94404, United States.
ACS Med Chem Lett ; 11(3): 358-364, 2020 Mar 12.
Article in En | MEDLINE | ID: mdl-32184970

Full text: 1 Collection: 01-internacional Database: MEDLINE Type of study: Prognostic_studies Language: En Journal: ACS Med Chem Lett Year: 2020 Type: Article Affiliation country: United States

Full text: 1 Collection: 01-internacional Database: MEDLINE Type of study: Prognostic_studies Language: En Journal: ACS Med Chem Lett Year: 2020 Type: Article Affiliation country: United States