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Synthesis of novel halogenated triarylpyrazoles as selective COX-2 inhibitors: Anti-inflammatory activity, histopatholgical profile and in-silico studies.
Abdellatif, Khaled R A; Abdelall, Eman K A; Labib, Madlen B; Fadaly, Wael A A; Zidan, Taha H.
Affiliation
  • Abdellatif KRA; Department of Pharmaceutical Organic Chemistry, Faculty of Pharmacy, Beni-Suef University, Beni-Suef 62514, Egypt; Department of Pharmaceutical Sciences, Ibn Sina National College for Medical Studies, Jeddah, Saudi Arabia.
  • Abdelall EKA; Department of Pharmaceutical Organic Chemistry, Faculty of Pharmacy, Beni-Suef University, Beni-Suef 62514, Egypt.
  • Labib MB; Department of Pharmaceutical Organic Chemistry, Faculty of Pharmacy, Beni-Suef University, Beni-Suef 62514, Egypt. Electronic address: madlen.wanas@pharm.bsu.edu.eg.
  • Fadaly WAA; Department of Pharmaceutical Organic Chemistry, Faculty of Pharmacy, Beni-Suef University, Beni-Suef 62514, Egypt.
  • Zidan TH; Department of Pharmaceutical Organic Chemistry, Faculty of Pharmacy, Beni-Suef University, Beni-Suef 62514, Egypt.
Bioorg Chem ; 105: 104418, 2020 12.
Article in En | MEDLINE | ID: mdl-33166844

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Pyrazoles / Anti-Inflammatory Agents, Non-Steroidal / Edema / Cyclooxygenase 2 / Cyclooxygenase 2 Inhibitors / Hydrocarbons, Halogenated Limits: Animals / Humans Language: En Journal: Bioorg Chem Year: 2020 Type: Article Affiliation country: Saudi Arabia

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Pyrazoles / Anti-Inflammatory Agents, Non-Steroidal / Edema / Cyclooxygenase 2 / Cyclooxygenase 2 Inhibitors / Hydrocarbons, Halogenated Limits: Animals / Humans Language: En Journal: Bioorg Chem Year: 2020 Type: Article Affiliation country: Saudi Arabia