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α-naphthoflavone-derived cytochrome P450 (CYP)1B1 degraders specific for sensitizing CYP1B1-mediated drug resistance to prostate cancer DU145: Structure activity relationship.
Chen, Peng; Wang, Shaobing; Cao, Chenyang; Ye, Wenchong; Wang, Meizhu; Zhou, Cui; Chen, Wenming; Zhang, Xu; Zhang, Keyu; Zhou, Wen.
Affiliation
  • Chen P; School of Pharmaceutical Sciences, Guangzhou University of Chinese Medicine, University town, Waihuan Rd., Panyu, Guangzhou, 510006, China; Shanghai Veterinary Research Institute, Chinese Academy of Agricultural Sciences, 200241, Shanghai, China.
  • Wang S; School of Pharmaceutical Sciences, South-Central University for nationalities, Wuhan, 430074, China.
  • Cao C; School of Pharmaceutical Sciences, Guangzhou University of Chinese Medicine, University town, Waihuan Rd., Panyu, Guangzhou, 510006, China.
  • Ye W; School of Pharmaceutical Sciences, Guangzhou University of Chinese Medicine, University town, Waihuan Rd., Panyu, Guangzhou, 510006, China.
  • Wang M; School of Pharmaceutical Sciences, Guangzhou University of Chinese Medicine, University town, Waihuan Rd., Panyu, Guangzhou, 510006, China.
  • Zhou C; School of Pharmaceutical Sciences, Guangzhou University of Chinese Medicine, University town, Waihuan Rd., Panyu, Guangzhou, 510006, China.
  • Chen W; Department of Pharmaceutical Production Center &TCM and Ethnomedicine Development International Laboratory, The First Hospital of Hunan University of Chinese Medicine, 95, Shaoshan Rd, Changsha, Hunan, 41007, China.
  • Zhang X; College of Forestry and Landscape Architecture, South China Agricultural University, 510642, China. Electronic address: zhangxu@126.com.
  • Zhang K; Shanghai Veterinary Research Institute, Chinese Academy of Agricultural Sciences, 200241, Shanghai, China; Key Laboratory of Veterinary Chemical Drugs and Pharmaceutics, Ministry of Agriculture and Rural Affairs, Shanghai Veterinary Research Institute, Chinese Academy of Agricultural Sciences, Shang
  • Zhou W; Shanghai Veterinary Research Institute, Chinese Academy of Agricultural Sciences, 200241, Shanghai, China; Key Laboratory of Veterinary Chemical Drugs and Pharmaceutics, Ministry of Agriculture and Rural Affairs, Shanghai Veterinary Research Institute, Chinese Academy of Agricultural Sciences, Shang
Bioorg Chem ; 116: 105295, 2021 11.
Article in En | MEDLINE | ID: mdl-34455300

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Prostatic Neoplasms / Benzoflavones / Drug Resistance, Neoplasm / Cytochrome P-450 CYP1B1 / Antineoplastic Agents Limits: Humans / Male Language: En Journal: Bioorg Chem Year: 2021 Type: Article Affiliation country: China

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Prostatic Neoplasms / Benzoflavones / Drug Resistance, Neoplasm / Cytochrome P-450 CYP1B1 / Antineoplastic Agents Limits: Humans / Male Language: En Journal: Bioorg Chem Year: 2021 Type: Article Affiliation country: China