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Thalidomide derivatives as nanomolar human neutrophil elastase inhibitors: Rational design, synthesis, antiproliferative activity and mechanism of action.
Donarska, Beata; Slawinska-Brych, Adrianna; Mizerska-Kowalska, Magdalena; Zdzisinska, Barbara; Plazinski, Wojciech; Laczkowski, Krzysztof Z.
Affiliation
  • Donarska B; Department of Chemical Technology and Pharmaceuticals, Faculty of Pharmacy, Collegium Medicum, Nicolaus Copernicus University, Jurasza 2, 85-089 Bydgoszcz, Poland. Electronic address: 265000@stud.umk.pl.
  • Slawinska-Brych A; Department of Cell Biology, Institute of Biological Sciences, Maria Curie-Sklodowska University, Akademicka 19 Street, 20-033 Lublin, Poland.
  • Mizerska-Kowalska M; Department of Virology and Immunology, Institute of Biological Sciences, Maria Curie-Sklodowska University, Akademicka 19 Street, 20-033 Lublin, Poland.
  • Zdzisinska B; Department of Virology and Immunology, Institute of Biological Sciences, Maria Curie-Sklodowska University, Akademicka 19 Street, 20-033 Lublin, Poland.
  • Plazinski W; Jerzy Haber Institute of Catalysis and Surface Chemistry, Polish Academy of Sciences, Niezapominajek 8, 30-239, Cracow, Poland; Department of Biopharmacy, Medical University of Lublin, Chodzki 4a, 20-093 Lublin, Poland.
  • Laczkowski KZ; Department of Chemical Technology and Pharmaceuticals, Faculty of Pharmacy, Collegium Medicum, Nicolaus Copernicus University, Jurasza 2, 85-089 Bydgoszcz, Poland.
Bioorg Chem ; 138: 106608, 2023 09.
Article in En | MEDLINE | ID: mdl-37207596

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Carcinoma, Non-Small-Cell Lung / Lung Neoplasms / Antineoplastic Agents Limits: Humans Language: En Journal: Bioorg Chem Year: 2023 Type: Article

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Carcinoma, Non-Small-Cell Lung / Lung Neoplasms / Antineoplastic Agents Limits: Humans Language: En Journal: Bioorg Chem Year: 2023 Type: Article