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Mutate and Conjugate: A Method to Enable Rapid In-Cell Target Validation.
Thomas, Adam M; Serafini, Marta; Grant, Emma K; Coombs, Edward A J; Bluck, Joseph P; Schiedel, Matthias; McDonough, Michael A; Reynolds, Jessica K; Lee, Bernadette; Platt, Michael; Sharlandjieva, Vassilena; Biggin, Philip C; Duarte, Fernanda; Milne, Thomas A; Bush, Jacob T; Conway, Stuart J.
Affiliation
  • Thomas AM; Department of Chemistry, Chemistry Research Laboratory, University of Oxford, Mansfield Road, Oxford OX1 3TA, United Kingdom.
  • Serafini M; Department of Chemistry, Chemistry Research Laboratory, University of Oxford, Mansfield Road, Oxford OX1 3TA, United Kingdom.
  • Grant EK; Department of Chemical Biology, GSK, Gunnels Wood Road, Stevenage, Hertfordshire SG1 2NY, United Kingdom.
  • Coombs EAJ; Department of Chemistry, Chemistry Research Laboratory, University of Oxford, Mansfield Road, Oxford OX1 3TA, United Kingdom.
  • Bluck JP; Department of Chemistry, Chemistry Research Laboratory, University of Oxford, Mansfield Road, Oxford OX1 3TA, United Kingdom.
  • Schiedel M; Department of Biochemistry, South Parks Road, Oxford OX1 3QU, United Kingdom.
  • McDonough MA; Department of Chemistry, Chemistry Research Laboratory, University of Oxford, Mansfield Road, Oxford OX1 3TA, United Kingdom.
  • Reynolds JK; Department of Chemistry, Chemistry Research Laboratory, University of Oxford, Mansfield Road, Oxford OX1 3TA, United Kingdom.
  • Lee B; Department of Chemistry, Chemistry Research Laboratory, University of Oxford, Mansfield Road, Oxford OX1 3TA, United Kingdom.
  • Platt M; Department of Chemistry, Chemistry Research Laboratory, University of Oxford, Mansfield Road, Oxford OX1 3TA, United Kingdom.
  • Sharlandjieva V; Department of Chemistry, Chemistry Research Laboratory, University of Oxford, Mansfield Road, Oxford OX1 3TA, United Kingdom.
  • Biggin PC; MRC Molecular Haematology Unit, MRC Weatherall Institute of Molecular Medicine, Radcliffe Department of Medicine, University of Oxford, Oxford OX3 9DS, United Kingdom.
  • Duarte F; Department of Biochemistry, South Parks Road, Oxford OX1 3QU, United Kingdom.
  • Milne TA; Department of Chemistry, Chemistry Research Laboratory, University of Oxford, Mansfield Road, Oxford OX1 3TA, United Kingdom.
  • Bush JT; MRC Molecular Haematology Unit, MRC Weatherall Institute of Molecular Medicine, Radcliffe Department of Medicine, University of Oxford, Oxford OX3 9DS, United Kingdom.
  • Conway SJ; Department of Chemical Biology, GSK, Gunnels Wood Road, Stevenage, Hertfordshire SG1 2NY, United Kingdom.
ACS Chem Biol ; 18(11): 2405-2417, 2023 11 17.
Article in En | MEDLINE | ID: mdl-37874862

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Transcription Factors / Nuclear Proteins Limits: Humans Language: En Journal: ACS Chem Biol Year: 2023 Type: Article Affiliation country: United kingdom

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Transcription Factors / Nuclear Proteins Limits: Humans Language: En Journal: ACS Chem Biol Year: 2023 Type: Article Affiliation country: United kingdom