Synthesis of 2-amido-2,3-dihydro-1H-phenalene derivatives as new conformationally restricted ligands for melatonin receptors.

Mathé-Allainmat, M; Gaudy, F; Sicsic, S; Dangy-Caye, A L; Shen, S; Brémont, B; Benatalah, Z; Langlois, M; Renard, P; Delagrange, P

Mathé-Allainmat, M; Gaudy, F; Sicsic, S; Dangy-Caye, A L; Shen, S; Brémont, B; Benatalah, Z; Langlois, M; Renard, P; Delagrange, P.

Affiliation

Mathé-Allainmat M; CNRS-BIOCIS, URA 1843, Faculté de Pharmacie, Châtenay-Malabry, France.

J Med Chem ; 39(16): 3089-95, 1996 Aug 02.

Article in En | MEDLINE | ID: mdl-8759629

Subject(s)

Amides/chemical synthesis; Melanocytes/drug effects; Polycyclic Compounds/chemical synthesis; Receptors, Cell Surface/agonists; Receptors, Cell Surface/metabolism; Amides/chemistry; Amides/metabolism; Amides/pharmacology; Animals; Ligands; Magnetic Resonance Spectroscopy; Melanocytes/physiology; Melanophores/drug effects; Melatonin/metabolism; Molecular Conformation; Molecular Structure; Polycyclic Compounds/chemistry; Polycyclic Compounds/metabolism; Polycyclic Compounds/pharmacology; Receptors, Melatonin; Structure-Activity Relationship; Xenopus laevis

Search on Google

XML

PubMed Links

Collection: 01-internacional Database: MEDLINE Main subject: Polycyclic Compounds / Receptors, Cell Surface / Amides / Melanocytes Limits: Animals Language: En Journal: J Med Chem Journal subject: QUIMICA Year: 1996 Type: Article Affiliation country: France

Search on Google

XML

PubMed Links