Development of 2,4-diaminopyrimidine derivatives as novel SNSR4 antagonists.
Bioorg Med Chem Lett
; 21(7): 2102-5, 2011 Apr 01.
Article
en En
| MEDLINE
| ID: mdl-21333534
ABSTRACT
2,4-Diaminopyrimidines derivatives were developed as a novel class of SNSR4 antagonists. Structure activity relationship of the diamino pyrimidine core was explored and a tool compound suitable for target validation was identified.
Texto completo:
1
Colección:
01-internacional
Banco de datos:
MEDLINE
Asunto principal:
Pirimidinas
/
Células Receptoras Sensoriales
/
Receptores de Superficie Celular
Idioma:
En
Revista:
Bioorg Med Chem Lett
Asunto de la revista:
BIOQUIMICA
/
QUIMICA
Año:
2011
Tipo del documento:
Article