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Discovery of thienopyrimidine-based FLT3 inhibitors from the structural modification of known IKKß inhibitors.
Park, Chun-Ho; Lee, Chulho; Yang, Jee Sun; Joe, Bo-Young; Chun, Kwangwoo; Kim, Hyuntae; Kim, Hye Yun; Kang, Jong Soon; Lee, Jangik I; Kim, Myung-Hwa; Han, Gyoonhee.
Afiliación
  • Park CH; Graduate Program in Biomaterials Science & Engineering, Yonsei University, Seodaemun-gu, Seoul 120-749, Republic of Korea; Division of New Drug Development, R&D Center, Jeil Pharmaceutical Co., Ltd 117-1, Keungok-Ri, Baekam-Myun, Cheoin-Gu, Yongin-City, Kyunggi-Do 449-861, Republic of Korea.
  • Lee C; Translational Research Center for Protein Function Control, Department of Biotechnology, Yonsei University, Seodaemun-gu, Seoul 120-749, Republic of Korea.
  • Yang JS; Translational Research Center for Protein Function Control, Department of Biotechnology, Yonsei University, Seodaemun-gu, Seoul 120-749, Republic of Korea.
  • Joe BY; Division of New Drug Development, R&D Center, Jeil Pharmaceutical Co., Ltd 117-1, Keungok-Ri, Baekam-Myun, Cheoin-Gu, Yongin-City, Kyunggi-Do 449-861, Republic of Korea.
  • Chun K; Division of New Drug Development, R&D Center, Jeil Pharmaceutical Co., Ltd 117-1, Keungok-Ri, Baekam-Myun, Cheoin-Gu, Yongin-City, Kyunggi-Do 449-861, Republic of Korea.
  • Kim H; Translational Research Center for Protein Function Control, Department of Biotechnology, Yonsei University, Seodaemun-gu, Seoul 120-749, Republic of Korea; Department of Biomedical Sciences (WCU Program), Yonsei University, Seodaemun-gu, Seoul 120-749, Republic of Korea.
  • Kim HY; Center for Neuro-Medicine of Brain Science Institute, Korea Institute of Science and Technology, Hwarangno 14-gil 5, Seongbuk-gu, Seoul 136-791, Republic of Korea.
  • Kang JS; Bioevaluation Center, Korea Research Institute of Bioscience and Biotechnology, Ochang, Cheongwon, Chungbuk 363-883, Republic of Korea.
  • Lee JI; College of Pharmacy, Yonsei University, 85 Songdogwahak-ro, Yeonsu-gu, Incheon 406-840, Republic of Korea.
  • Kim MH; Division of New Drug Development, R&D Center, Jeil Pharmaceutical Co., Ltd 117-1, Keungok-Ri, Baekam-Myun, Cheoin-Gu, Yongin-City, Kyunggi-Do 449-861, Republic of Korea. Electronic address: mhkim@kddf.org.
  • Han G; Translational Research Center for Protein Function Control, Department of Biotechnology, Yonsei University, Seodaemun-gu, Seoul 120-749, Republic of Korea; Department of Biomedical Sciences (WCU Program), Yonsei University, Seodaemun-gu, Seoul 120-749, Republic of Korea. Electronic address: gyoonhee
Bioorg Med Chem Lett ; 24(12): 2655-60, 2014 Jun 15.
Article en En | MEDLINE | ID: mdl-24813730

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Pirimidinas / Quinasa I-kappa B / Tirosina Quinasa 3 Similar a fms / Bibliotecas de Moléculas Pequeñas Límite: Humans Idioma: En Revista: Bioorg Med Chem Lett Asunto de la revista: BIOQUIMICA / QUIMICA Año: 2014 Tipo del documento: Article

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Pirimidinas / Quinasa I-kappa B / Tirosina Quinasa 3 Similar a fms / Bibliotecas de Moléculas Pequeñas Límite: Humans Idioma: En Revista: Bioorg Med Chem Lett Asunto de la revista: BIOQUIMICA / QUIMICA Año: 2014 Tipo del documento: Article