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A Molecular Dynamics Investigation of Mycobacterium tuberculosis Prenyl Synthases: Conformational Flexibility and Implications for Computer-aided Drug Discovery.
Kim, Meekyum Olivia; Feng, Xinxin; Feixas, Ferran; Zhu, Wei; Lindert, Steffen; Bogue, Shannon; Sinko, William; de Oliveira, César; Rao, Guodong; Oldfield, Eric; McCammon, James Andrew.
Afiliación
  • Kim MO; Department of Chemistry and Biochemistry, University of California San Diego, La Jolla, CA, 92093, USA.
  • Feng X; Department of Chemistry, University of Illinois at Urbana-Champaign, Urbana, IL, 61801, USA.
  • Feixas F; Department of Pharmacology, University of California San Diego, La Jolla, CA, 92093, USA.
  • Zhu W; Department of Chemistry, University of Illinois at Urbana-Champaign, Urbana, IL, 61801, USA.
  • Lindert S; Department of Pharmacology, University of California San Diego, La Jolla, CA, 92093, USA.
  • Bogue S; Howard Hughes Medical Institute, University of California San Diego, La Jolla, CA, 92093, USA.
  • Sinko W; Department of Chemistry, University of Illinois at Urbana-Champaign, Urbana, IL, 61801, USA.
  • de Oliveira C; Department of Pharmacology, University of California San Diego, La Jolla, CA, 92093, USA.
  • Rao G; Department of Chemistry and Biochemistry, University of California San Diego, La Jolla, CA, 92093, USA.
  • Oldfield E; Department of Pharmacology, University of California San Diego, La Jolla, CA, 92093, USA.
  • McCammon JA; Howard Hughes Medical Institute, University of California San Diego, La Jolla, CA, 92093, USA.
Chem Biol Drug Des ; 85(6): 756-69, 2015 Jun.
Article en En | MEDLINE | ID: mdl-25352216

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Transferasas Alquil y Aril / Inhibidores Enzimáticos / Geraniltranstransferasa / Mycobacterium tuberculosis / Antituberculosos Tipo de estudio: Prognostic_studies Límite: Humans Idioma: En Revista: Chem Biol Drug Des Asunto de la revista: BIOQUIMICA / FARMACIA / FARMACOLOGIA Año: 2015 Tipo del documento: Article País de afiliación: Estados Unidos

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Transferasas Alquil y Aril / Inhibidores Enzimáticos / Geraniltranstransferasa / Mycobacterium tuberculosis / Antituberculosos Tipo de estudio: Prognostic_studies Límite: Humans Idioma: En Revista: Chem Biol Drug Des Asunto de la revista: BIOQUIMICA / FARMACIA / FARMACOLOGIA Año: 2015 Tipo del documento: Article País de afiliación: Estados Unidos