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Inhibition of AMP-Activated Protein Kinase at the Allosteric Drug-Binding Site Promotes Islet Insulin Release.
Scott, John W; Galic, Sandra; Graham, Kate L; Foitzik, Richard; Ling, Naomi X Y; Dite, Toby A; Issa, Samah M A; Langendorf, Chris G; Weng, Qing Ping; Thomas, Helen E; Kay, Thomas W; Birnberg, Neal C; Steinberg, Gregory R; Kemp, Bruce E; Oakhill, Jonathan S.
Afiliación
  • Scott JW; Protein Chemistry & Metabolism Unit, St Vincent's Institute of Medical Research and Department of Medicine, University of Melbourne, 41 Victoria Parade, Fitzroy, VIC 3065, Australia. Electronic address: jscott@svi.edu.au.
  • Galic S; Protein Chemistry & Metabolism Unit, St Vincent's Institute of Medical Research and Department of Medicine, University of Melbourne, 41 Victoria Parade, Fitzroy, VIC 3065, Australia.
  • Graham KL; Immunology and Diabetes Unit, St Vincent's Institute of Medical Research, 41 Victoria Parade, Fitzroy, VIC 3065, Australia.
  • Foitzik R; Cancer Therapeutics CRC Pty Ltd, Medicinal Chemistry and Drug Action, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, VIC 3052, Australia.
  • Ling NX; Protein Chemistry & Metabolism Unit, St Vincent's Institute of Medical Research and Department of Medicine, University of Melbourne, 41 Victoria Parade, Fitzroy, VIC 3065, Australia.
  • Dite TA; Protein Chemistry & Metabolism Unit, St Vincent's Institute of Medical Research and Department of Medicine, University of Melbourne, 41 Victoria Parade, Fitzroy, VIC 3065, Australia.
  • Issa SM; Protein Chemistry & Metabolism Unit, St Vincent's Institute of Medical Research and Department of Medicine, University of Melbourne, 41 Victoria Parade, Fitzroy, VIC 3065, Australia.
  • Langendorf CG; Protein Chemistry & Metabolism Unit, St Vincent's Institute of Medical Research and Department of Medicine, University of Melbourne, 41 Victoria Parade, Fitzroy, VIC 3065, Australia.
  • Weng QP; Mercury Therapeutics Inc., 175 East New Boston Street, Woburn, MA 01801, USA.
  • Thomas HE; Immunology and Diabetes Unit, St Vincent's Institute of Medical Research, 41 Victoria Parade, Fitzroy, VIC 3065, Australia.
  • Kay TW; Immunology and Diabetes Unit, St Vincent's Institute of Medical Research, 41 Victoria Parade, Fitzroy, VIC 3065, Australia.
  • Birnberg NC; Mercury Therapeutics Inc., 175 East New Boston Street, Woburn, MA 01801, USA.
  • Steinberg GR; Division of Endocrinology and Metabolism, Department of Medicine, McMaster University, 1200 Main Street West, Hamilton, ON L8N 3Z5, Canada.
  • Kemp BE; Protein Chemistry & Metabolism Unit, St Vincent's Institute of Medical Research and Department of Medicine, University of Melbourne, 41 Victoria Parade, Fitzroy, VIC 3065, Australia.
  • Oakhill JS; Protein Chemistry & Metabolism Unit, St Vincent's Institute of Medical Research and Department of Medicine, University of Melbourne, 41 Victoria Parade, Fitzroy, VIC 3065, Australia. Electronic address: joakhill@svi.edu.au.
Chem Biol ; 22(6): 705-11, 2015 Jun 18.
Article en En | MEDLINE | ID: mdl-26091167

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Proteínas Quinasas Activadas por AMP / Hidroxiquinolinas / Insulina Límite: Animals / Humans Idioma: En Revista: Chem Biol Asunto de la revista: BIOLOGIA / BIOQUIMICA / QUIMICA Año: 2015 Tipo del documento: Article

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Proteínas Quinasas Activadas por AMP / Hidroxiquinolinas / Insulina Límite: Animals / Humans Idioma: En Revista: Chem Biol Asunto de la revista: BIOLOGIA / BIOQUIMICA / QUIMICA Año: 2015 Tipo del documento: Article