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2,8-Disubstituted-1,6-Naphthyridines and 4,6-Disubstituted-Isoquinolines with Potent, Selective Affinity for CDK8/19.
Mallinger, Aurélie; Schiemann, Kai; Rink, Christian; Sejberg, Jimmy; Honey, Mark A; Czodrowski, Paul; Stubbs, Mark; Poeschke, Oliver; Busch, Michael; Schneider, Richard; Schwarz, Daniel; Musil, Djordje; Burke, Rosemary; Urbahns, Klaus; Workman, Paul; Wienke, Dirk; Clarke, Paul A; Raynaud, Florence I; Eccles, Suzanne A; Esdar, Christina; Rohdich, Felix; Blagg, Julian.
Afiliación
  • Mallinger A; Cancer Research UK Cancer Therapeutics Unit, The Institute of Cancer Research , London SW7 3RP, UK.
  • Schiemann K; Merck KGaA, Darmstadt 64293, Germany.
  • Rink C; Cancer Research UK Cancer Therapeutics Unit, The Institute of Cancer Research , London SW7 3RP, UK.
  • Sejberg J; Cancer Research UK Cancer Therapeutics Unit, The Institute of Cancer Research , London SW7 3RP, UK.
  • Honey MA; Cancer Research UK Cancer Therapeutics Unit, The Institute of Cancer Research , London SW7 3RP, UK.
  • Czodrowski P; Merck KGaA, Darmstadt 64293, Germany.
  • Stubbs M; Cancer Research UK Cancer Therapeutics Unit, The Institute of Cancer Research , London SW7 3RP, UK.
  • Poeschke O; Merck KGaA, Darmstadt 64293, Germany.
  • Busch M; Merck KGaA, Darmstadt 64293, Germany.
  • Schneider R; Merck KGaA, Darmstadt 64293, Germany.
  • Schwarz D; Merck KGaA, Darmstadt 64293, Germany.
  • Musil D; Merck KGaA, Darmstadt 64293, Germany.
  • Burke R; Cancer Research UK Cancer Therapeutics Unit, The Institute of Cancer Research , London SW7 3RP, UK.
  • Urbahns K; Merck KGaA, Darmstadt 64293, Germany.
  • Workman P; Cancer Research UK Cancer Therapeutics Unit, The Institute of Cancer Research , London SW7 3RP, UK.
  • Wienke D; Merck KGaA, Darmstadt 64293, Germany.
  • Clarke PA; Cancer Research UK Cancer Therapeutics Unit, The Institute of Cancer Research , London SW7 3RP, UK.
  • Raynaud FI; Cancer Research UK Cancer Therapeutics Unit, The Institute of Cancer Research , London SW7 3RP, UK.
  • Eccles SA; Cancer Research UK Cancer Therapeutics Unit, The Institute of Cancer Research , London SW7 3RP, UK.
  • Esdar C; Merck KGaA, Darmstadt 64293, Germany.
  • Rohdich F; Merck KGaA, Darmstadt 64293, Germany.
  • Blagg J; Cancer Research UK Cancer Therapeutics Unit, The Institute of Cancer Research , London SW7 3RP, UK.
ACS Med Chem Lett ; 7(6): 573-8, 2016 Jun 09.
Article en En | MEDLINE | ID: mdl-27326329

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Idioma: En Revista: ACS Med Chem Lett Año: 2016 Tipo del documento: Article País de afiliación: Reino Unido

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Idioma: En Revista: ACS Med Chem Lett Año: 2016 Tipo del documento: Article País de afiliación: Reino Unido