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Crystal structures of human glycine receptor α3 bound to a novel class of analgesic potentiators.
Huang, Xin; Shaffer, Paul L; Ayube, Shawn; Bregman, Howard; Chen, Hao; Lehto, Sonya G; Luther, Jason A; Matson, David J; McDonough, Stefan I; Michelsen, Klaus; Plant, Matthew H; Schneider, Stephen; Simard, Jeffrey R; Teffera, Yohannes; Yi, Shuyan; Zhang, Maosheng; DiMauro, Erin F; Gingras, Jacinthe.
Afiliación
  • Huang X; Department of Molecular Structure and Characterization, Amgen Inc., Cambridge, Massachusetts, USA.
  • Shaffer PL; Department of Molecular Structure and Characterization, Amgen Inc., Cambridge, Massachusetts, USA.
  • Ayube S; Department of Molecular Structure and Characterization, Amgen Inc., Cambridge, Massachusetts, USA.
  • Bregman H; Department of Medicinal Chemistry, Amgen Inc., Cambridge, Massachusetts, USA.
  • Chen H; Department of Protein Technologies, Amgen Inc., Cambridge, Massachusetts, USA.
  • Lehto SG; Department of Neuroscience, Amgen Inc., Thousand Oaks, California, USA.
  • Luther JA; Department of Neuroscience, Amgen Inc., Cambridge, Massachusetts, USA.
  • Matson DJ; Department of Neuroscience, Amgen Inc., Cambridge, Massachusetts, USA.
  • McDonough SI; Department of Neuroscience, Amgen Inc., Cambridge, Massachusetts, USA.
  • Michelsen K; Department of Discovery Attribute Sciences, Amgen Inc., Cambridge, Massachusetts, USA.
  • Plant MH; Department of Discovery Attribute Sciences, Amgen Inc., Cambridge, Massachusetts, USA.
  • Schneider S; Department of Neuroscience, Amgen Inc., Cambridge, Massachusetts, USA.
  • Simard JR; Department of Neuroscience, Amgen Inc., Cambridge, Massachusetts, USA.
  • Teffera Y; Department of Pharmacokinetics &Drug Metabolism, Amgen Inc., Cambridge, Massachusetts, USA.
  • Yi S; Department of Medicinal Chemistry, Amgen Inc., Cambridge, Massachusetts, USA.
  • Zhang M; Department of Neuroscience, Amgen Inc., Thousand Oaks, California, USA.
  • DiMauro EF; Department of Medicinal Chemistry, Amgen Inc., Cambridge, Massachusetts, USA.
  • Gingras J; Department of Neuroscience, Amgen Inc., Cambridge, Massachusetts, USA.
Nat Struct Mol Biol ; 24(2): 108-113, 2017 02.
Article en En | MEDLINE | ID: mdl-27991902

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Receptores de Glicina Límite: Humans Idioma: En Revista: Nat Struct Mol Biol Asunto de la revista: BIOLOGIA MOLECULAR Año: 2017 Tipo del documento: Article País de afiliación: Estados Unidos

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Receptores de Glicina Límite: Humans Idioma: En Revista: Nat Struct Mol Biol Asunto de la revista: BIOLOGIA MOLECULAR Año: 2017 Tipo del documento: Article País de afiliación: Estados Unidos