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Identification of 5-(1-Methyl-5-(trifluoromethyl)-1H-pyrazol-3-yl)thiophene-2-Carboxamides as Novel and Selective Monoamine Oxidase B Inhibitors Used to Improve Memory and Cognition.
Kaplan, Alan P; Keenan, Terence; Scott, Roderick; Zhou, Xianbo; Bourchouladze, Rusiko; McRiner, Andrew J; Wilson, Mark E; Romashko, Darlene; Miller, Regina; Bletsch, Matthew; Anderson, Gary; Stanley, Jennifer; Zhang, Adia; Lee, Dong; Nikpur, John.
Afiliación
  • Kaplan AP; Dart NeuroScience, LLC , 12278 Scripps Summit Drive, San Diego, California 92131, United States.
  • Keenan T; Dart NeuroScience, LLC , 12278 Scripps Summit Drive, San Diego, California 92131, United States.
  • Scott R; Dart NeuroScience, LLC , 12278 Scripps Summit Drive, San Diego, California 92131, United States.
  • Zhou X; SJN Biomed LTD , 398 West Second Ring Road, Kunming 650118, China.
  • Bourchouladze R; Dart NeuroScience, LLC , 12278 Scripps Summit Drive, San Diego, California 92131, United States.
  • McRiner AJ; X-Chem Pharmaceuticals, Inc. , 100 Beaver Street, Suite 101, Waltham, Massachusetts 02453, United States.
  • Wilson ME; Dart NeuroScience, LLC , 12278 Scripps Summit Drive, San Diego, California 92131, United States.
  • Romashko D; Aset Therapeutics , 25 Health Sciences Drive, Stony Brook, New York 11790, United States.
  • Miller R; Bristol-Myers Squibb , 5 Research Parkway, Wallingford, Connecticut 06492, United States.
  • Bletsch M; The Hain Celestial Group , 1111 Marcus Avenue, New Hyde Park, New York 11042, United States.
  • Anderson G; Dart NeuroScience, LLC , 12278 Scripps Summit Drive, San Diego, California 92131, United States.
  • Stanley J; Dart NeuroScience, LLC , 12278 Scripps Summit Drive, San Diego, California 92131, United States.
  • Zhang A; Dart NeuroScience, LLC , 12278 Scripps Summit Drive, San Diego, California 92131, United States.
  • Lee D; Dart NeuroScience, LLC , 12278 Scripps Summit Drive, San Diego, California 92131, United States.
  • Nikpur J; Dart NeuroScience, LLC , 12278 Scripps Summit Drive, San Diego, California 92131, United States.
ACS Chem Neurosci ; 8(12): 2746-2758, 2017 12 20.
Article en En | MEDLINE | ID: mdl-28857544

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Ácidos Carboxílicos / Cognición / Nootrópicos / Memoria / Monoaminooxidasa Tipo de estudio: Diagnostic_studies / Observational_studies / Prognostic_studies Límite: Animals Idioma: En Revista: ACS Chem Neurosci Año: 2017 Tipo del documento: Article País de afiliación: Estados Unidos

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Ácidos Carboxílicos / Cognición / Nootrópicos / Memoria / Monoaminooxidasa Tipo de estudio: Diagnostic_studies / Observational_studies / Prognostic_studies Límite: Animals Idioma: En Revista: ACS Chem Neurosci Año: 2017 Tipo del documento: Article País de afiliación: Estados Unidos