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Multisite phosphorylation is required for sustained interaction with GRKs and arrestins during rapid µ-opioid receptor desensitization.
Miess, Elke; Gondin, Arisbel B; Yousuf, Arsalan; Steinborn, Ralph; Mösslein, Nadja; Yang, Yunshi; Göldner, Martin; Ruland, Julia G; Bünemann, Moritz; Krasel, Cornelius; Christie, MacDonald J; Halls, Michelle L; Schulz, Stefan; Canals, Meritxell.
Afiliación
  • Miess E; Department of Pharmacology and Toxicology, Jena University Hospital-Friedrich Schiller University Jena, D-07747 Jena, Germany.
  • Gondin AB; Drug Discovery Biology Theme, Monash Institute of Pharmaceutical Sciences, Monash University, Victoria 3052, Australia.
  • Yousuf A; Discipline of Pharmacology, University of Sydney, New South Wales 2006, Australia.
  • Steinborn R; Department of Pharmacology and Toxicology, Jena University Hospital-Friedrich Schiller University Jena, D-07747 Jena, Germany.
  • Mösslein N; Department of Pharmacology and Toxicology, Philipps-University Marburg, D-35043 Marburg, Germany.
  • Yang Y; Department of Pharmacology and Toxicology, Philipps-University Marburg, D-35043 Marburg, Germany.
  • Göldner M; Department of Pharmacology and Toxicology, Philipps-University Marburg, D-35043 Marburg, Germany.
  • Ruland JG; Department of Pharmacology and Toxicology, Philipps-University Marburg, D-35043 Marburg, Germany.
  • Bünemann M; Department of Pharmacology and Toxicology, Philipps-University Marburg, D-35043 Marburg, Germany.
  • Krasel C; Department of Pharmacology and Toxicology, Philipps-University Marburg, D-35043 Marburg, Germany.
  • Christie MJ; Discipline of Pharmacology, University of Sydney, New South Wales 2006, Australia.
  • Halls ML; Drug Discovery Biology Theme, Monash Institute of Pharmaceutical Sciences, Monash University, Victoria 3052, Australia.
  • Schulz S; Department of Pharmacology and Toxicology, Jena University Hospital-Friedrich Schiller University Jena, D-07747 Jena, Germany. stefan.schulz@med.uni-jena.de meri.canals@monash.edu.
  • Canals M; Drug Discovery Biology Theme, Monash Institute of Pharmaceutical Sciences, Monash University, Victoria 3052, Australia. stefan.schulz@med.uni-jena.de meri.canals@monash.edu.
Sci Signal ; 11(539)2018 07 17.
Article en En | MEDLINE | ID: mdl-30018083

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Regulación de la Expresión Génica / Receptores Opioides mu / Arrestinas / Encefalina Ala(2)-MeFe(4)-Gli(5) / Quinasa 2 del Receptor Acoplado a Proteína-G Tipo de estudio: Prognostic_studies Límite: Humans Idioma: En Revista: Sci Signal Asunto de la revista: CIENCIA / FISIOLOGIA Año: 2018 Tipo del documento: Article País de afiliación: Alemania

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Regulación de la Expresión Génica / Receptores Opioides mu / Arrestinas / Encefalina Ala(2)-MeFe(4)-Gli(5) / Quinasa 2 del Receptor Acoplado a Proteína-G Tipo de estudio: Prognostic_studies Límite: Humans Idioma: En Revista: Sci Signal Asunto de la revista: CIENCIA / FISIOLOGIA Año: 2018 Tipo del documento: Article País de afiliación: Alemania