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α-Helix-Mimicking Sulfono-γ-AApeptide Inhibitors for p53-MDM2/MDMX Protein-Protein Interactions.
Sang, Peng; Shi, Yan; Lu, Junhao; Chen, Lihong; Yang, Leixiang; Borcherds, Wade; Abdulkadir, Sami; Li, Qi; Daughdrill, Gary; Chen, Jiandong; Cai, Jianfeng.
Afiliación
  • Sang P; Department of Chemistry , University of South Florida , 4202 E. Fowler Avenue , Tampa , Florida 33620 , United States.
  • Shi Y; Department of Chemistry , University of South Florida , 4202 E. Fowler Avenue , Tampa , Florida 33620 , United States.
  • Lu J; Department of Molecular Oncology , H. Lee Moffitt Cancer Center and Research Institute , 12902 Magnolia Drive , Tampa , Florida 33612 , United States.
  • Chen L; Department of Molecular Oncology , H. Lee Moffitt Cancer Center and Research Institute , 12902 Magnolia Drive , Tampa , Florida 33612 , United States.
  • Yang L; Department of Molecular Oncology , H. Lee Moffitt Cancer Center and Research Institute , 12902 Magnolia Drive , Tampa , Florida 33612 , United States.
  • Borcherds W; Department of Cell Biology, Microbiology and Molecular Biology , University of South Florida , Tampa , Florida 33620 , United States.
  • Abdulkadir S; Department of Chemistry , University of South Florida , 4202 E. Fowler Avenue , Tampa , Florida 33620 , United States.
  • Li Q; Department of Medical Oncology , Shuguang Hospital, Shanghai University of Traditional Chinese Medicine , Shanghai 201203 , China.
  • Daughdrill G; Department of Cell Biology, Microbiology and Molecular Biology , University of South Florida , Tampa , Florida 33620 , United States.
  • Chen J; Department of Molecular Oncology , H. Lee Moffitt Cancer Center and Research Institute , 12902 Magnolia Drive , Tampa , Florida 33612 , United States.
  • Cai J; Department of Chemistry , University of South Florida , 4202 E. Fowler Avenue , Tampa , Florida 33620 , United States.
J Med Chem ; 63(3): 975-986, 2020 02 13.
Article en En | MEDLINE | ID: mdl-31971801

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Unión Proteica / Sulfonas / Proteína p53 Supresora de Tumor / Proteínas Proto-Oncogénicas / Proteínas de Ciclo Celular / Proteínas Proto-Oncogénicas c-mdm2 / Peptidomiméticos Límite: Humans Idioma: En Revista: J Med Chem Asunto de la revista: QUIMICA Año: 2020 Tipo del documento: Article País de afiliación: Estados Unidos

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Unión Proteica / Sulfonas / Proteína p53 Supresora de Tumor / Proteínas Proto-Oncogénicas / Proteínas de Ciclo Celular / Proteínas Proto-Oncogénicas c-mdm2 / Peptidomiméticos Límite: Humans Idioma: En Revista: J Med Chem Asunto de la revista: QUIMICA Año: 2020 Tipo del documento: Article País de afiliación: Estados Unidos