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Preclinical Safety Assessment of a Highly Selective and Potent Dual Small-Molecule Inhibitor of CBP/P300 in Rats and Dogs.
Katavolos, Paula; Cain, Gary; Farman, Cindy; Romero, F Anthony; Magnuson, Steven; Ly, Justin Q; Choo, Edna F; Katakam, Anand Kumar; Andaya, Roxanne; Maher, Jonathan.
Afiliación
  • Katavolos P; Safety Assessment, Genentech, Inc, South San Francisco, CA, USA.
  • Cain G; Safety Assessment, Genentech, Inc, South San Francisco, CA, USA.
  • Farman C; Safety Assessment, Genentech, Inc, South San Francisco, CA, USA.
  • Romero FA; Vet Path Services, Inc, Mason, OH, USA.
  • Magnuson S; Medicinal Chemistry, Genentech, Inc, South San Francisco, CA, USA.
  • Ly JQ; Terns Pharmaceuticals, San Mateo, CA, USA.
  • Choo EF; Medicinal Chemistry, Genentech, Inc, South San Francisco, CA, USA.
  • Katakam AK; Department of Drug Metabolism and Pharmacology, Genentech, Inc, South San Francisco, CA, USA.
  • Andaya R; Department of Drug Metabolism and Pharmacology, Genentech, Inc, South San Francisco, CA, USA.
  • Maher J; Department of Pathology, Genentech, Inc, South San Francisco, CA USA.
Toxicol Pathol ; 48(3): 465-480, 2020 04.
Article en En | MEDLINE | ID: mdl-32124659

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Pirazoles / Piridinas / Factores de Transcripción p300-CBP Tipo de estudio: Prognostic_studies Límite: Animals / Female / Humans / Male Idioma: En Revista: Toxicol Pathol Año: 2020 Tipo del documento: Article País de afiliación: Estados Unidos

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Pirazoles / Piridinas / Factores de Transcripción p300-CBP Tipo de estudio: Prognostic_studies Límite: Animals / Female / Humans / Male Idioma: En Revista: Toxicol Pathol Año: 2020 Tipo del documento: Article País de afiliación: Estados Unidos