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6,7-Dimethoxy-2-phenethyl-1,2,3,4-tetrahydroisoquinoline amides and corresponding ester isosteres as multidrug resistance reversers.
Braconi, Laura; Bartolucci, Gianluca; Contino, Marialessandra; Chiaramonte, Niccolò; Giampietro, Roberta; Manetti, Dina; Perrone, Maria Grazia; Romanelli, Maria Novella; Colabufo, Nicola Antonio; Riganti, Chiara; Dei, Silvia; Teodori, Elisabetta.
Afiliación
  • Braconi L; NEUROFARBA Department, Section of Pharmaceutical and Nutraceutical Sciences, University of Florence, Florence, Italy.
  • Bartolucci G; NEUROFARBA Department, Section of Pharmaceutical and Nutraceutical Sciences, University of Florence, Florence, Italy.
  • Contino M; Department of Pharmacy-Drug Sciences, University of Bari "A. Moro", Bari, Italy.
  • Chiaramonte N; NEUROFARBA Department, Section of Pharmaceutical and Nutraceutical Sciences, University of Florence, Florence, Italy.
  • Giampietro R; Department of Pharmacy-Drug Sciences, University of Bari "A. Moro", Bari, Italy.
  • Manetti D; NEUROFARBA Department, Section of Pharmaceutical and Nutraceutical Sciences, University of Florence, Florence, Italy.
  • Perrone MG; Department of Pharmacy-Drug Sciences, University of Bari "A. Moro", Bari, Italy.
  • Romanelli MN; NEUROFARBA Department, Section of Pharmaceutical and Nutraceutical Sciences, University of Florence, Florence, Italy.
  • Colabufo NA; Department of Pharmacy-Drug Sciences, University of Bari "A. Moro", Bari, Italy.
  • Riganti C; Department of Oncology, University of Turin, Turin, Italy.
  • Dei S; NEUROFARBA Department, Section of Pharmaceutical and Nutraceutical Sciences, University of Florence, Florence, Italy.
  • Teodori E; NEUROFARBA Department, Section of Pharmaceutical and Nutraceutical Sciences, University of Florence, Florence, Italy.
J Enzyme Inhib Med Chem ; 35(1): 974-992, 2020 Dec.
Article en En | MEDLINE | ID: mdl-32253945

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Resistencia a Múltiples Medicamentos / Resistencia a Antineoplásicos / Tetrahidroisoquinolinas / Ésteres / Amidas / Neoplasias / Antineoplásicos Límite: Animals / Humans Idioma: En Revista: J Enzyme Inhib Med Chem Asunto de la revista: BIOQUIMICA / QUIMICA Año: 2020 Tipo del documento: Article País de afiliación: Italia

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Resistencia a Múltiples Medicamentos / Resistencia a Antineoplásicos / Tetrahidroisoquinolinas / Ésteres / Amidas / Neoplasias / Antineoplásicos Límite: Animals / Humans Idioma: En Revista: J Enzyme Inhib Med Chem Asunto de la revista: BIOQUIMICA / QUIMICA Año: 2020 Tipo del documento: Article País de afiliación: Italia