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Single Peptide Backbone Surrogate Mutations to Regulate Angiotensin GPCR Subtype Selectivity.
Vrettos, Eirinaios I; Valverde, Ibai E; Mascarin, Alba; Pallier, Patrick N; Cerofolini, Linda; Fragai, Marco; Parigi, Giacomo; Hirmiz, Baydaa; Bekas, Nick; Grob, Nathalie M; Stylos, Evgenios Κ; Shaye, Hamidreza; Del Borgo, Mark; Aguilar, Marie-Isabel; Magnani, Francesca; Syed, Nelofer; Crook, Timothy; Waqif, Emal; Ghazaly, Essam; Cherezov, Vadim; Widdop, Robert E; Luchinat, Claudio; Michael-Titus, Adina T; Mindt, Thomas L; Tzakos, Andreas G.
Afiliación
  • Vrettos EI; Department of Chemistry, University of Ioannina, Ioannina, 45110, Greece.
  • Valverde IE; Division of Radiopharmaceutical Chemistry, University of Basel Hospital, Petersgraben 4, 4031, Basel, Switzerland.
  • Mascarin A; Institut de Chimie Moléculaire de l'Université de Bourgogne (ICMUB), UMR 6302 CNRS, Université de Bourgogne Franche-Comté, 9 Avenue Alain Savary, 21000, Dijon, France.
  • Pallier PN; Division of Radiopharmaceutical Chemistry, University of Basel Hospital, Petersgraben 4, 4031, Basel, Switzerland.
  • Cerofolini L; Centre for Neuroscience and Trauma, The Blizard Institute, Barts and The London School of Medicine and Dentistry, Queen Mary, University of London, 4 Newark Street, Whitechapel, London, E1 2AT, UK.
  • Fragai M; Consorzio Interuniversitario Risonanze Magnetiche MetalloProteine, (CIRMMP), University of Florence, Sesto Fiorentino, 50019, Italy.
  • Parigi G; Centre for Magnetic Resonance, CERM, University of Florence, Sesto Fiorentino, 50019, Italy.
  • Hirmiz B; Consorzio Interuniversitario Risonanze Magnetiche MetalloProteine, (CIRMMP), University of Florence, Sesto Fiorentino, 50019, Italy.
  • Bekas N; Centre for Magnetic Resonance, CERM, University of Florence, Sesto Fiorentino, 50019, Italy.
  • Grob NM; Consorzio Interuniversitario Risonanze Magnetiche MetalloProteine, (CIRMMP), University of Florence, Sesto Fiorentino, 50019, Italy.
  • Stylos EΚ; Monash Biomedicine Discovery Institute and Department of Biochemistry, and Molecular Biology, Monash University, Clayton, VIC, 3800, Australia.
  • Shaye H; Department of Chemistry, University of Ioannina, Ioannina, 45110, Greece.
  • Del Borgo M; Department of Chemistry and Applied Biosciences, ETH Zurich, 8093, Zürich, Switzerland.
  • Aguilar MI; Department of Chemistry, University of Ioannina, Ioannina, 45110, Greece.
  • Magnani F; Bridge Institute, Department of Chemistry, University of Southern California., Los Angeles, CA, 90089, USA.
  • Syed N; Monash Biomedicine Discovery Institute and Department of Biochemistry, and Molecular Biology, Monash University, Clayton, VIC, 3800, Australia.
  • Crook T; Monash Biomedicine Discovery Institute and Department of Biochemistry, and Molecular Biology, Monash University, Clayton, VIC, 3800, Australia.
  • Waqif E; Department of Biology and Biotechnology "Lazzaro Spallanzani", University of Pavia, Pavia, Italy.
  • Ghazaly E; John Fulcher Neuro-oncology Laboratory, Division of Brain Sciences, Faculty of Medicine, Imperial College London, London, W6 8RP, UK.
  • Cherezov V; Leaders in Oncology Care, 95 Harley Street, London, W1G 6AF, UK.
  • Widdop RE; Centre for Neuroscience and Trauma, The Blizard Institute, Barts and The London School of Medicine and Dentistry, Queen Mary, University of London, 4 Newark Street, Whitechapel, London, E1 2AT, UK.
  • Luchinat C; Centre for Haemato-Oncology, Barts Cancer Institute, Queen Mary University of London, London, UK.
  • Michael-Titus AT; Bridge Institute, Department of Chemistry, University of Southern California., Los Angeles, CA, 90089, USA.
  • Mindt TL; Monash Biomedicine Discovery Institute and Department of Pharmacology, Monash University, Clayton, VIC, 3800, Australia.
  • Tzakos AG; Centre for Magnetic Resonance, CERM, University of Florence, Sesto Fiorentino, 50019, Italy.
Chemistry ; 26(47): 10690-10694, 2020 Aug 21.
Article en En | MEDLINE | ID: mdl-32691857

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Péptidos / Angiotensina II / Receptores de Angiotensina / Mutación Límite: Animals / Humans Idioma: En Revista: Chemistry Asunto de la revista: QUIMICA Año: 2020 Tipo del documento: Article País de afiliación: Grecia

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Péptidos / Angiotensina II / Receptores de Angiotensina / Mutación Límite: Animals / Humans Idioma: En Revista: Chemistry Asunto de la revista: QUIMICA Año: 2020 Tipo del documento: Article País de afiliación: Grecia