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The structural basis for high affinity binding of α1-acid glycoprotein to the potent antitumor compound UCN-01.
Landin, Erik J B; Williams, Christopher; Ryan, Sara A; Bochel, Alice; Akter, Nahida; Redfield, Christina; Sessions, Richard B; Dedi, Neesha; Taylor, Richard J; Crump, Matthew P.
Afiliación
  • Landin EJB; School of Chemistry, University of Bristol, Bristol, UK.
  • Williams C; School of Chemistry, University of Bristol, Bristol, UK; BrisSynBio, University of Bristol, Bristol, UK.
  • Ryan SA; School of Chemistry, University of Bristol, Bristol, UK.
  • Bochel A; School of Chemistry, University of Bristol, Bristol, UK.
  • Akter N; School of Chemistry, University of Bristol, Bristol, UK.
  • Redfield C; Department of Biochemistry, University of Oxford, Oxford, UK.
  • Sessions RB; School of Biochemistry, University of Bristol, Bristol, UK.
  • Dedi N; Discovery Sciences, UCB Biopharma, Slough, UK.
  • Taylor RJ; Discovery Sciences, UCB Biopharma, Slough, UK. Electronic address: Richard.taylor@ucb.com.
  • Crump MP; School of Chemistry, University of Bristol, Bristol, UK. Electronic address: matt.crump@bristol.ac.uk.
J Biol Chem ; 297(6): 101392, 2021 12.
Article en En | MEDLINE | ID: mdl-34758357

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Orosomucoide / Estaurosporina / Antineoplásicos Límite: Humans Idioma: En Revista: J Biol Chem Año: 2021 Tipo del documento: Article País de afiliación: Reino Unido

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Orosomucoide / Estaurosporina / Antineoplásicos Límite: Humans Idioma: En Revista: J Biol Chem Año: 2021 Tipo del documento: Article País de afiliación: Reino Unido