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Structural and Molecular Insight into Piperazine and Piperidine Derivatives as Histamine H3 and Sigma-1 Receptor Antagonists with Promising Antinociceptive Properties.
Szczepanska, Katarzyna; Podlewska, Sabina; Dichiara, Maria; Gentile, Davide; Patamia, Vincenzo; Rosier, Niklas; Mönnich, Denise; Ruiz Cantero, Ma Carmen; Karcz, Tadeusz; Lazewska, Dorota; Siwek, Agata; Pockes, Steffen; Cobos, Enrique J; Marrazzo, Agostino; Stark, Holger; Rescifina, Antonio; Bojarski, Andrzej J; Amata, Emanuele; Kiec-Kononowicz, Katarzyna.
Afiliación
  • Szczepanska K; Department of Technology and Biotechnology of Drugs, Faculty of Pharmacy, Jagiellonian University Medical College, Medyczna 9, Kraków 30-688, Poland.
  • Podlewska S; Maj Institute of Pharmacology, Polish Academy of Sciences, Smetna 12, Kraków 31-343, Poland.
  • Dichiara M; Department of Technology and Biotechnology of Drugs, Faculty of Pharmacy, Jagiellonian University Medical College, Medyczna 9, Kraków 30-688, Poland.
  • Gentile D; Maj Institute of Pharmacology, Polish Academy of Sciences, Smetna 12, Kraków 31-343, Poland.
  • Patamia V; Department of Drug and Health Sciences, University of Catania, V.le A. Doria, 95125 Catania, Italy.
  • Rosier N; Department of Drug and Health Sciences, University of Catania, V.le A. Doria, 95125 Catania, Italy.
  • Mönnich D; Department of Drug and Health Sciences, University of Catania, V.le A. Doria, 95125 Catania, Italy.
  • Ruiz Cantero MC; Institute of Pharmacy, Faculty of Chemistry and Pharmacy, University of Regensburg, Universitätsstraße 31, D-93053 Regensburg, Germany.
  • Karcz T; Institute of Pharmacy, Faculty of Chemistry and Pharmacy, University of Regensburg, Universitätsstraße 31, D-93053 Regensburg, Germany.
  • Lazewska D; Department of Pharmacology and Neurosciences Institute (Biomedical Research Center) and Biosanitary Research Institute ibs.GRANADA, University of Granada, Avenida de la Investigación 11, 18016 Granada, Spain.
  • Siwek A; Department of Technology and Biotechnology of Drugs, Faculty of Pharmacy, Jagiellonian University Medical College, Medyczna 9, Kraków 30-688, Poland.
  • Pockes S; Department of Technology and Biotechnology of Drugs, Faculty of Pharmacy, Jagiellonian University Medical College, Medyczna 9, Kraków 30-688, Poland.
  • Cobos EJ; Department of Pharmacobiology, Faculty of Pharmacy, Jagiellonian University Medical College, Medyczna 9, Kraków 30-688, Poland.
  • Marrazzo A; Institute of Pharmacy, Faculty of Chemistry and Pharmacy, University of Regensburg, Universitätsstraße 31, D-93053 Regensburg, Germany.
  • Stark H; Department of Pharmacology and Neurosciences Institute (Biomedical Research Center) and Biosanitary Research Institute ibs.GRANADA, University of Granada, Avenida de la Investigación 11, 18016 Granada, Spain.
  • Rescifina A; Department of Drug and Health Sciences, University of Catania, V.le A. Doria, 95125 Catania, Italy.
  • Bojarski AJ; Institute of Pharmaceutical and Medicinal Chemistry, Heinrich Heine University Düsseldorf, Universitaetsstr. 1, 40225 Duesseldorf, Germany.
  • Amata E; Department of Drug and Health Sciences, University of Catania, V.le A. Doria, 95125 Catania, Italy.
  • Kiec-Kononowicz K; Maj Institute of Pharmacology, Polish Academy of Sciences, Smetna 12, Kraków 31-343, Poland.
ACS Chem Neurosci ; 13(1): 1-15, 2022 01 05.
Article en En | MEDLINE | ID: mdl-34908391

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Receptores Histamínicos H3 / Antagonistas de los Receptores Histamínicos H3 Idioma: En Revista: ACS Chem Neurosci Año: 2022 Tipo del documento: Article País de afiliación: Polonia

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Receptores Histamínicos H3 / Antagonistas de los Receptores Histamínicos H3 Idioma: En Revista: ACS Chem Neurosci Año: 2022 Tipo del documento: Article País de afiliación: Polonia