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Discovery of MK-1454: A Potent Cyclic Dinucleotide Stimulator of Interferon Genes Agonist for the Treatment of Cancer.
Chang, Wonsuk; Altman, Michael D; Lesburg, Charles A; Perera, Samanthi A; Piesvaux, Jennifer A; Schroeder, Gottfried K; Wyss, Daniel F; Cemerski, Saso; Chen, Yiping; DiNunzio, Edward; Haidle, Andrew M; Ho, Thu; Kariv, Ilona; Knemeyer, Ian; Kopinja, Johnny E; Lacey, Brian M; Laskey, Jason; Lim, Jongwon; Long, Brian J; Ma, Yanhong; Maddess, Matthew L; Pan, Bo-Sheng; Presland, Jeremy P; Spooner, Edward; Steinhuebel, Dietrich; Truong, Quang; Zhang, Zhibo; Fu, Jianmin; Addona, George H; Northrup, Alan B; Parmee, Emma; Tata, James R; Bennett, David Jonathan; Cumming, Jared N; Siu, Tony; Trotter, B Wesley.
Afiliación
  • Chang W; Merck & Co., Inc., Kenilworth, New Jersey 07033, United States.
  • Altman MD; Merck & Co., Inc., Boston, Massachusetts 02115, United States.
  • Lesburg CA; Merck & Co., Inc., Boston, Massachusetts 02115, United States.
  • Perera SA; Merck & Co., Inc., Boston, Massachusetts 02115, United States.
  • Piesvaux JA; Merck & Co., Inc., Boston, Massachusetts 02115, United States.
  • Schroeder GK; Merck & Co., Inc., Boston, Massachusetts 02115, United States.
  • Wyss DF; Merck & Co., Inc., Kenilworth, New Jersey 07033, United States.
  • Cemerski S; Merck & Co., Inc., Boston, Massachusetts 02115, United States.
  • Chen Y; Merck & Co., Inc., Boston, Massachusetts 02115, United States.
  • DiNunzio E; Merck & Co., Inc., Kenilworth, New Jersey 07033, United States.
  • Haidle AM; Merck & Co., Inc., Boston, Massachusetts 02115, United States.
  • Ho T; Merck & Co., Inc., West Point, Pennsylvania 19486, United States.
  • Kariv I; Merck & Co., Inc., Boston, Massachusetts 02115, United States.
  • Knemeyer I; Merck & Co., Inc., Boston, Massachusetts 02115, United States.
  • Kopinja JE; Merck & Co., Inc., Boston, Massachusetts 02115, United States.
  • Lacey BM; Merck & Co., Inc., Boston, Massachusetts 02115, United States.
  • Laskey J; Merck & Co., Inc., Boston, Massachusetts 02115, United States.
  • Lim J; Merck & Co., Inc., Boston, Massachusetts 02115, United States.
  • Long BJ; Merck & Co., Inc., Boston, Massachusetts 02115, United States.
  • Ma Y; Merck & Co., Inc., Boston, Massachusetts 02115, United States.
  • Maddess ML; Merck & Co., Inc., Boston, Massachusetts 02115, United States.
  • Pan BS; Merck & Co., Inc., Boston, Massachusetts 02115, United States.
  • Presland JP; Merck & Co., Inc., Boston, Massachusetts 02115, United States.
  • Spooner E; Merck & Co., Inc., Boston, Massachusetts 02115, United States.
  • Steinhuebel D; Merck & Co., Inc., Boston, Massachusetts 02115, United States.
  • Truong Q; Merck & Co., Inc., Kenilworth, New Jersey 07033, United States.
  • Zhang Z; Pharmaron Beijing Co. Ltd., Beijing 100176, P. R. China.
  • Fu J; Pharmaron Beijing Co. Ltd., Beijing 100176, P. R. China.
  • Addona GH; Merck & Co., Inc., Boston, Massachusetts 02115, United States.
  • Northrup AB; Merck & Co., Inc., Boston, Massachusetts 02115, United States.
  • Parmee E; Merck & Co., Inc., Kenilworth, New Jersey 07033, United States.
  • Tata JR; Merck & Co., Inc., Kenilworth, New Jersey 07033, United States.
  • Bennett DJ; Merck & Co., Inc., Boston, Massachusetts 02115, United States.
  • Cumming JN; Merck & Co., Inc., Boston, Massachusetts 02115, United States.
  • Siu T; Merck & Co., Inc., Boston, Massachusetts 02115, United States.
  • Trotter BW; Merck & Co., Inc., Boston, Massachusetts 02115, United States.
J Med Chem ; 65(7): 5675-5689, 2022 04 14.
Article en En | MEDLINE | ID: mdl-35332774

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Proteínas de la Membrana / Neoplasias Límite: Animals / Humans Idioma: En Revista: J Med Chem Asunto de la revista: QUIMICA Año: 2022 Tipo del documento: Article País de afiliación: Estados Unidos

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Proteínas de la Membrana / Neoplasias Límite: Animals / Humans Idioma: En Revista: J Med Chem Asunto de la revista: QUIMICA Año: 2022 Tipo del documento: Article País de afiliación: Estados Unidos