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Synthesis, In Vitro Biological Evaluation and In Silico Molecular Docking Studies of Indole Based Thiadiazole Derivatives as Dual Inhibitor of Acetylcholinesterase and Butyrylchloinesterase.
Khan, Shoaib; Iqbal, Shahid; Taha, Muhammad; Rahim, Fazal; Shah, Mazloom; Ullah, Hayat; Bahadur, Ali; Alrbyawi, Hamad; Dera, Ayed A; Alahmdi, Mohammed Issa; Pashameah, Rami Adel; Alzahrani, Eman; Farouk, Abd-ElAziem.
Afiliación
  • Khan S; Department of Chemistry, Hazara University, Mansehra 21120, Pakistan.
  • Iqbal S; Department of Chemistry, School of Natural Sciences (SNS), National University of Science and Technology (NUST), H-12, Islamabad 46000, Pakistan.
  • Taha M; Department of Clinical Pharmacy, Institute for Research and Medical Consultations (IRMC), Imam Abdulrah-Man Bin Faisal University, Dammam 34212, Saudi Arabia.
  • Rahim F; Department of Chemistry, Hazara University, Mansehra 21120, Pakistan.
  • Shah M; Department of Chemistry, Abbottabad University of Science and Technology (AUST), Abbottabad 22500, Pakistan.
  • Ullah H; Department of Chemistry, University of Okara, Okara 56300, Pakistan.
  • Bahadur A; Department of Chemistry, College of Science and Technology, Wenzhou-Kean University, Wenzhou 325060, China.
  • Alrbyawi H; Pharmaceutics and Pharmaceutical Technology Department, College of Pharmacy, Taibah University, Medina 42353, Saudi Arabia.
  • Dera AA; Department of Clinical Laboratory Sciences, College of Applied Medical Sciences, King Khalid University, Abha 61413, Saudi Arabia.
  • Alahmdi MI; Department of Chemistry, Faculty of Science, University of Tabuk, Tabuk 71491, Saudi Arabia.
  • Pashameah RA; Department of Chemistry, Faculty of Applied Science, Umm Al-Qura University, Makkah 24230, Saudi Arabia.
  • Alzahrani E; Department of Chemistry, College of Science, Taif University, Taif 21944, Saudi Arabia.
  • Farouk AE; Department of Biotechnology, College of Science, Taif University, Taif 21944, Saudi Arabia.
Molecules ; 27(21)2022 Oct 29.
Article en En | MEDLINE | ID: mdl-36364195

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Acetilcolinesterasa / Tiadiazoles Idioma: En Revista: Molecules Asunto de la revista: BIOLOGIA Año: 2022 Tipo del documento: Article País de afiliación: Pakistán

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Acetilcolinesterasa / Tiadiazoles Idioma: En Revista: Molecules Asunto de la revista: BIOLOGIA Año: 2022 Tipo del documento: Article País de afiliación: Pakistán