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Design, synthesis and antitumor activity of novel thiophene- triazine derivatives bearing arylurea unit as potent PI3K/mTOR inhibitorss.
Xu, Shan; Luo, Leixuan; Sun, Xin; Yang, Yang; Guo, Qiuyan; Jiang, Zhiyan; Wu, Yingliang.
Afiliación
  • Xu S; Department of Pharmacology, Shenyang Pharmaceutical University, 103, Wenhua Road, Shenhe District, Shenyang 110016, China; Jiangxi Provincial Key Laboratory of Drug Design and Evaluation, School of Pharmacy, Jiangxi Science & Technology Normal University, 605, Fenglin Road, Nanchang, Jiangxi 330
  • Luo L; Jiangxi Provincial Key Laboratory of Drug Design and Evaluation, School of Pharmacy, Jiangxi Science & Technology Normal University, 605, Fenglin Road, Nanchang, Jiangxi 330013, China.
  • Sun X; Jiangxi Provincial Key Laboratory of Drug Design and Evaluation, School of Pharmacy, Jiangxi Science & Technology Normal University, 605, Fenglin Road, Nanchang, Jiangxi 330013, China.
  • Yang Y; Jiangxi Provincial Key Laboratory of Drug Design and Evaluation, School of Pharmacy, Jiangxi Science & Technology Normal University, 605, Fenglin Road, Nanchang, Jiangxi 330013, China.
  • Guo Q; Jiangxi Provincial Key Laboratory of Drug Design and Evaluation, School of Pharmacy, Jiangxi Science & Technology Normal University, 605, Fenglin Road, Nanchang, Jiangxi 330013, China.
  • Jiang Z; Jiangxi Provincial Key Laboratory of Drug Design and Evaluation, School of Pharmacy, Jiangxi Science & Technology Normal University, 605, Fenglin Road, Nanchang, Jiangxi 330013, China.
  • Wu Y; Department of Pharmacology, Shenyang Pharmaceutical University, 103, Wenhua Road, Shenhe District, Shenyang 110016, China. Electronic address: yingliang_1016@163.com.
Bioorg Med Chem ; 78: 117133, 2023 01 15.
Article en En | MEDLINE | ID: mdl-36599263

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Fosfatidilinositol 3-Quinasas / Antineoplásicos Límite: Humans Idioma: En Revista: Bioorg Med Chem Asunto de la revista: BIOQUIMICA / QUIMICA Año: 2023 Tipo del documento: Article

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Fosfatidilinositol 3-Quinasas / Antineoplásicos Límite: Humans Idioma: En Revista: Bioorg Med Chem Asunto de la revista: BIOQUIMICA / QUIMICA Año: 2023 Tipo del documento: Article