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Ugi reaction-assisted assembly of covalent PROTACs against glutathione peroxidase 4.
Zhu, Liquan; Hu, Shiqi; Yan, Xiaoqiao; Zeng, Qian; Zhang, Bei; Jiang, Linye; Yao, Shao Q; Ge, Jingyan.
Afiliación
  • Zhu L; Key Laboratory of Bioorganic Synthesis of Zhejiang Province, College of Biotechnology and Bioengineering, Zhejiang University of Technology, Hangzhou 310014, PR China.
  • Hu S; Key Laboratory of Bioorganic Synthesis of Zhejiang Province, College of Biotechnology and Bioengineering, Zhejiang University of Technology, Hangzhou 310014, PR China.
  • Yan X; Key Laboratory of Bioorganic Synthesis of Zhejiang Province, College of Biotechnology and Bioengineering, Zhejiang University of Technology, Hangzhou 310014, PR China.
  • Zeng Q; Key Laboratory of Bioorganic Synthesis of Zhejiang Province, College of Biotechnology and Bioengineering, Zhejiang University of Technology, Hangzhou 310014, PR China.
  • Zhang B; Key Laboratory of Bioorganic Synthesis of Zhejiang Province, College of Biotechnology and Bioengineering, Zhejiang University of Technology, Hangzhou 310014, PR China.
  • Jiang L; Key Laboratory of Bioorganic Synthesis of Zhejiang Province, College of Biotechnology and Bioengineering, Zhejiang University of Technology, Hangzhou 310014, PR China.
  • Yao SQ; Department of Chemistry, National University of Singapore, 4 Science Drive 2, Singapore 117544, Singapore. Electronic address: chmyaosq@nus.edu.sg.
  • Ge J; Key Laboratory of Bioorganic Synthesis of Zhejiang Province, College of Biotechnology and Bioengineering, Zhejiang University of Technology, Hangzhou 310014, PR China. Electronic address: gejy@zjut.edu.cn.
Bioorg Chem ; 134: 106461, 2023 05.
Article en En | MEDLINE | ID: mdl-36924654

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Quimera Dirigida a la Proteólisis Idioma: En Revista: Bioorg Chem Año: 2023 Tipo del documento: Article

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Quimera Dirigida a la Proteólisis Idioma: En Revista: Bioorg Chem Año: 2023 Tipo del documento: Article