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Optimization of a Class of Dihydrobenzofurane Analogs toward Orally Efficacious YAP-TEAD Protein-Protein Interaction Inhibitors.
Sellner, Holger; Chapeau, Emilie; Furet, Pascal; Voegtle, Markus; Salem, Bahaa; Le Douget, Mickaël; Bordas, Vincent; Groell, Jean-Marc; Le Goff, Anne-Laure; Rouzet, Christine; Wietlisbach, Thomas; Zimmermann, Thomas; McKenna, Joseph; Brocklehurst, Cara E; Chène, Patrick; Wartmann, Markus; Scheufler, Clemens; Kallen, Joerg; Williams, Gareth; Harlfinger, Stephanie; Traebert, Martin; Dumotier, Bérengère M; Schmelzle, Tobias; Soldermann, Nicolas.
Afiliación
  • Sellner H; Global Discovery Chemistry, Novartis Institutes for BioMedical Research, Basel, 4002, Switzerland.
  • Chapeau E; Oncology Drug Discovery, Novartis Institutes for BioMedical Research, Basel, 4002, Switzerland.
  • Furet P; Global Discovery Chemistry, Novartis Institutes for BioMedical Research, Basel, 4002, Switzerland.
  • Voegtle M; Global Discovery Chemistry, Novartis Institutes for BioMedical Research, Basel, 4002, Switzerland.
  • Salem B; Global Discovery Chemistry, Novartis Institutes for BioMedical Research, Basel, 4002, Switzerland.
  • Le Douget M; Global Discovery Chemistry, Novartis Institutes for BioMedical Research, Basel, 4002, Switzerland.
  • Bordas V; Global Discovery Chemistry, Novartis Institutes for BioMedical Research, Basel, 4002, Switzerland.
  • Groell JM; Global Discovery Chemistry, Novartis Institutes for BioMedical Research, Basel, 4002, Switzerland.
  • Le Goff AL; Global Discovery Chemistry, Novartis Institutes for BioMedical Research, Basel, 4002, Switzerland.
  • Rouzet C; Global Discovery Chemistry, Novartis Institutes for BioMedical Research, Basel, 4002, Switzerland.
  • Wietlisbach T; Global Discovery Chemistry, Novartis Institutes for BioMedical Research, Basel, 4002, Switzerland.
  • Zimmermann T; Global Discovery Chemistry, Novartis Institutes for BioMedical Research, Basel, 4002, Switzerland.
  • McKenna J; Global Discovery Chemistry, Novartis Institutes for BioMedical Research, Basel, 4002, Switzerland.
  • Brocklehurst CE; Global Discovery Chemistry, Novartis Institutes for BioMedical Research, Basel, 4002, Switzerland.
  • Chène P; Oncology Drug Discovery, Novartis Institutes for BioMedical Research, Basel, 4002, Switzerland.
  • Wartmann M; Oncology Drug Discovery, Novartis Institutes for BioMedical Research, Basel, 4002, Switzerland.
  • Scheufler C; Chemical Biology & Therapeutics, Novartis Institutes for BioMedical Research, Basel, 4002, Switzerland.
  • Kallen J; Chemical Biology & Therapeutics, Novartis Institutes for BioMedical Research, Basel, 4002, Switzerland.
  • Williams G; Pharmacokinetics Sciences, Novartis Institutes for BioMedical Research, Basel, 4002, Switzerland.
  • Harlfinger S; Pharmacokinetics Sciences, Novartis Institutes for BioMedical Research, Basel, 4002, Switzerland.
  • Traebert M; Preclinical Safety, Novartis Institutes for BioMedical Research, Basel, 4002, Switzerland.
  • Dumotier BM; Preclinical Safety, Novartis Institutes for BioMedical Research, Basel, 4002, Switzerland.
  • Schmelzle T; Oncology Drug Discovery, Novartis Institutes for BioMedical Research, Basel, 4002, Switzerland.
  • Soldermann N; Global Discovery Chemistry, Novartis Institutes for BioMedical Research, Basel, 4002, Switzerland.
ChemMedChem ; 18(11): e202300051, 2023 06 01.
Article en En | MEDLINE | ID: mdl-36988034

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Factores de Transcripción / Neoplasias Tipo de estudio: Prognostic_studies Límite: Animals Idioma: En Revista: ChemMedChem Asunto de la revista: FARMACOLOGIA / QUIMICA Año: 2023 Tipo del documento: Article País de afiliación: Suiza

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Factores de Transcripción / Neoplasias Tipo de estudio: Prognostic_studies Límite: Animals Idioma: En Revista: ChemMedChem Asunto de la revista: FARMACOLOGIA / QUIMICA Año: 2023 Tipo del documento: Article País de afiliación: Suiza